SCHEMBL28042899

SCHEMBL28042899

Cn1ncc(I)c1CC(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 8/20 0.48
PTGDR2 Q9Y5Y4 2/20 0.33
ITGB3 P05106 1/20 0.32
ITGAV P06756 1/20 0.32
THRA P10827 1/20 0.32
THRB P10828 1/20 0.32
RXRA P19793 1/20 0.32
PPARG P37231 1/20 0.32
ALDH1A1 P00352 3/20 0.32
KDM4E B2RXH2 2/20 0.32
MAPT P10636 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
MAPK1 P28482 1/20 0.32
HPGD P15428 1/20 0.32
HSD17B10 Q99714 1/20 0.32
CYP3A4 P08684 1/20 0.32
GABRA1 P14867 1/20 0.32
TSHR P16473 1/20 0.32
NFKB1 P19838 1/20 0.32
GABRR1 P24046 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2777106 0.79 P2RX7 (0.47) P2RX7PTGDR2ALDH1A1KDM4EMAPK1
SCHEMBL4362725 0.79 PTGDR2 (0.38) P2RX7PTGDR2ALDH1A1KDM4EMAPT
SCHEMBL4361450 0.78 P2RX7 (0.51) P2RX7ALDH1A1MAPTHPGD
SCHEMBL16156183 0.78 MEN1 (0.38) ALDH1A1MAPTHPGD
SCHEMBL24044109 0.76 MAPK1 (0.39) P2RX7PTGDR2ALDH1A1KDM4EMAPT
SCHEMBL2594257 0.76
SCHEMBL12806714 0.74
SCHEMBL4359176 0.74 POLB (0.39) ALDH1A1KDM4EMAPTMAPK1HPGD
SCHEMBL24664567 0.74 PTGDR2 (0.33) P2RX7PTGDR2AGBL2LPAR1
SCHEMBL5410258 0.73 GAA (0.48) KDM4EL3MBTL1HPGDCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143203-A N-piperidin-3-ylbenzamide derivatives for the treatment of cardiovascular diseases PFIZER 2015-12-09 CN disclosed