SCHEMBL28042900

SCHEMBL28042900

Cln1ccc2ccncc21

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.53
MAPT P10636 15/20 0.47
CDC7 O00311 1/20 0.46
CDK2 P24941 1/20 0.46
SLC22A12 Q96S37 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27976818 0.87 CDC7 (0.45) CYP19A1MAPTCDC7CDK2SLC22A12
SCHEMBL3224575 0.74 CDC7 (0.50) CYP19A1MAPTCDC7CDK2
SCHEMBL18821827 0.74 CYP19A1 (0.49) CYP19A1MAPTCDC7CDK2
SCHEMBL10197253 0.74 CYP19A1 (0.49) CYP19A1MAPTCDC7CDK2
SCHEMBL29509135 0.74 MAPT (0.68) CYP19A1MAPTCDC7CDK2
SCHEMBL255050 0.74 MAPT (0.68) CYP19A1MAPTCDC7CDK2
SCHEMBL1892608 0.74 CYP19A1 (0.49) CYP19A1MAPTCDC7CDK2
SCHEMBL30768345 0.74 CYP19A1 (0.49) CYP19A1MAPTCDC7CDK2SLC22A12
SCHEMBL19190841 0.74 CYP19A1 (0.49) CYP19A1MAPTCDC7CDK2
SCHEMBL18822052 0.74 CYP19A1 (0.45) CYP19A1MAPTCDC7CDK2SLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105530932-B Primary formamide as BTK inhibitor 艾伯维公司 2019-09-27 CN disclosed
CN-106459042-B Anti-fibrotic pyridinones 英特穆恩公司 2019-06-28 CN disclosed
CN-109069481-A Methods and compounds for restoring function of mutant p53 皮姆维制药公司 2018-12-21 CN disclosed
CN-105143203-A N-piperidin-3-ylbenzamide derivatives for the treatment of cardiovascular diseases PFIZER 2015-12-09 CN disclosed