SCHEMBL28043326

SCHEMBL28043326

COc1cccc(-c2cc3cccnc3n2S(=O)(=O)c2ccccc2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC40A1 Q9NP59 2/20 0.47
GLO1 Q04760 1/20 0.47
HTR6 P50406 1/20 0.46
CYP2C19 P33261 1/20 0.46
MAPT P10636 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
MET P08581 1/20 0.44
CCNE1 P24864 2/20 0.44
CDK2 P24941 2/20 0.44
PDE4A P27815 4/20 0.43
PDE4B Q07343 4/20 0.43
PDE4C Q08493 4/20 0.43
PDE4D Q08499 4/20 0.43
TOP1 P11387 1/20 0.43
DYRK1A Q13627 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
ALDH1A1 P00352 2/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8126772 0.86 CYP2C19 (0.57) SLC40A1GLO1CYP2C19MAPTTDP1
SCHEMBL30405579 0.80 CYP2C19 (0.51) HTR6CYP2C19MAPTCCNE1CDK2
SCHEMBL5716751 0.80 PDE4A (0.46) SLC40A1CYP2C19MAPTCCNE1CDK2
SCHEMBL5716793 0.79 HDAC3 (0.55) SLC40A1GLO1CYP2C19MAPTTDP1
SCHEMBL31160496 0.76 L3MBTL1 (0.46) SLC40A1CYP2C19MAPTCCNE1CDK2
SCHEMBL30337641 0.75 CYP2C19 (0.56) SLC40A1GLO1HTR6CYP2C19MAPT
SCHEMBL1772416 0.75 CYP2C19 (0.56) SLC40A1GLO1HTR6CYP2C19MAPT
SCHEMBL1962059 0.74 HDAC3 (0.43) SLC40A1GLO1HTR6CYP2C19MAPT
SCHEMBL1962060 0.74 HDAC3 (0.43) SLC40A1GLO1HTR6CYP2C19MAPT
SCHEMBL5716795 0.74 CYP2C19 (0.42) SLC40A1CYP2C19MAPTCCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105246890-A Pyrrolo[2, 3-b]pyridine cdk9 kinase inhibitors ABBVIE INC 2016-01-13 CN disclosed