SCHEMBL28043907

SCHEMBL28043907

C=C(C(=O)OC(=O)c1cc(F)c([N+](=O)[O-])cc1F)C(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.41
ITGA5 P08648 1/20 0.41
ESPL1 Q14674 1/20 0.37
ALDH1A1 P00352 5/20 0.36
HIF1A Q16665 1/20 0.36
MAPT P10636 4/20 0.33
ATM Q13315 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
GPR174 Q9BXC1 1/20 0.33
HTT P42858 3/20 0.32
GPR35 Q9HC97 1/20 0.32
LMNA P02545 2/20 0.32
VCAM1 P19320 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
GAA P10253 1/20 0.31
THRB P10828 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CA1 P00915 1/20 0.31
MMP2 P08253 1/20 0.31
CA14 Q9ULX7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30041882 0.83 ITGB1 (0.47) ITGB1ITGA5ESPL1ALDH1A1HIF1A
SCHEMBL27552998 0.82 ALDH1A1 (0.41) ITGB1ITGA5ALDH1A1HIF1AMAPT
SCHEMBL27834939 0.81 TDP1 (0.42) ITGB1ITGA5ALDH1A1MAPTATM
SCHEMBL28824451 0.81 ATM (0.42) ITGB1ITGA5ALDH1A1HIF1AMAPT
SCHEMBL28791798 0.81 ITGB1 (0.51) ITGB1ITGA5ALDH1A1HIF1AMAPT
SCHEMBL16137955 0.79 ITGB1 (0.40) ITGB1ITGA5ESPL1ALDH1A1HIF1A
SCHEMBL28158467 0.78 TSHR (0.40) ITGB1ITGA5ALDH1A1MAPTTDP1
SCHEMBL1560111 0.77 PDGFRB (0.47) ITGB1ITGA5ESPL1ALDH1A1HIF1A
SCHEMBL27570720 0.77 ALDH1A1 (0.46) ITGB1ITGA5ALDH1A1MAPTHTT
SCHEMBL28270666 0.75 ITGB1 (0.38) ITGB1ITGA5ALDH1A1MAPTATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108164513-A Substituted oxo pyridine derivative and its purposes in terms of cardiovascular disorder is treated 拜耳制药股份公司 2018-06-15 CN disclosed
CN-105164122-A Substituted oxopyridine derivatives and their use in the treatment of cardiovascular disorders Bayer Pharma AG 2015-12-16 CN disclosed