SCHEMBL28043961

SCHEMBL28043961

Cc1cc(C)cc(-c2cc(NCCCCCN)nc(N)n2)c1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 12/20 0.54
TLR8 Q9NR97 6/20 0.53
HRH3 Q9Y5N1 1/20 0.41
AURKA O14965 1/20 0.41
JAK1 P23458 1/20 0.41
KDR P35968 1/20 0.41
SYK P43405 1/20 0.41
KCNH2 Q12809 1/20 0.41
LRRK2 Q5S007 1/20 0.41
AURKB Q96GD4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28151084 0.99 HRH4 (0.55) HRH4TLR8HRH3AURKAJAK1
SCHEMBL28043727 0.94 HRH4 (0.56) HRH4TLR8HRH3AURKASYK
SCHEMBL28151149 0.90 HRH4 (0.64) HRH4TLR8AURKAAURKB
SCHEMBL28043930 0.89 HRH4 (0.55) HRH4TLR8AURKAAURKB
SCHEMBL28267199 0.88 TLR8 (0.65) HRH4TLR8AURKAAURKB
SCHEMBL28152094 0.85 HRH4 (0.54) HRH4TLR8AURKAAURKB
SCHEMBL28845266 0.82 CYP2D6 (0.55) HRH4TLR8AURKAAURKB
SCHEMBL28267608 0.81 TLR8 (0.50) HRH4TLR8HRH3AURKAAURKB
SCHEMBL28267189 0.81 TLR8 (0.53) HRH4TLR8AURKAAURKB
SCHEMBL28845271 0.80 HRH4 (0.72) HRH4TLR8HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143206-B Pyrimidine -2,4- diamine derivative for treating cancer 托马斯·黑勒戴药物研究基金会 2019-01-15 CN disclosed
CN-105143206-A Pyrimidine-2,4-diamine derivatives for treatment of cancer THOMAS HELLEDAYS STIFTELSE F R MEDICINSK FORSKNING 2015-12-09 CN disclosed