SCHEMBL28267199

SCHEMBL28267199

CCCCCNc1cc(-c2cc(C)cc(C)c2)nc(N)n1

nearest known ligand 0.65

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 4/20 0.65
HRH4 Q9H3N8 9/20 0.51
AURKA O14965 1/20 0.41
PDPK1 O15530 1/20 0.41
TGFBR1 P36897 1/20 0.41
AURKB Q96GD4 1/20 0.41
DNM2 P50570 6/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28151084 0.89 HRH4 (0.55) TLR8HRH4AURKAPDPK1TGFBR1
SCHEMBL28151149 0.88 HRH4 (0.64) TLR8HRH4AURKAPDPK1TGFBR1
SCHEMBL28043961 0.88 HRH4 (0.54) TLR8HRH4AURKAAURKB
SCHEMBL28043727 0.87 HRH4 (0.56) TLR8HRH4AURKAPDPK1TGFBR1
SCHEMBL28043930 0.84 HRH4 (0.55) TLR8HRH4AURKAPDPK1TGFBR1
SCHEMBL28043772 0.84 AURKA (0.54) TLR8HRH4AURKAPDPK1TGFBR1
SCHEMBL28152094 0.83 HRH4 (0.54) TLR8HRH4AURKAPDPK1TGFBR1
SCHEMBL28845266 0.83 CYP2D6 (0.55) TLR8HRH4AURKAPDPK1TGFBR1
SCHEMBL28267189 0.82 TLR8 (0.53) TLR8HRH4AURKAPDPK1TGFBR1
SCHEMBL28267608 0.82 TLR8 (0.50) TLR8HRH4AURKAPDPK1TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143206-B Pyrimidine -2,4- diamine derivative for treating cancer 托马斯·黑勒戴药物研究基金会 2019-01-15 CN disclosed