SCHEMBL28044454

SCHEMBL28044454

O=[N+]([O-])c1ccc(OC2CCN([SH](=O)=O)CC2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.41
HTT P42858 1/20 0.41
RECQL P46063 1/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
MAPT P10636 3/20 0.40
POLB P06746 3/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HSPB1 P04792 1/20 0.38
KCNJ1 P48048 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11044966 0.82 EPHX2 (0.54) EPHX2SIGMAR1SMN1; SMN2CES2CES1
SCHEMBL28297004 0.82 SIGMAR1 (0.45) EPHX2SIGMAR1SMN1; SMN2HTTRECQL
SCHEMBL3274096 0.82 HRH3 (0.55) EPHX2SIGMAR1SMN1; SMN2HTTRECQL
SCHEMBL16532717 0.82 SIGMAR1 (0.45) EPHX2SIGMAR1SMN1; SMN2HTTRECQL
SCHEMBL4459795 0.81 CYP1A2 (0.52) EPHX2SIGMAR1CYP1A2CYP2D6KCNH2
SCHEMBL14626169 0.79 RECQL (0.46) EPHX2SIGMAR1SMN1; SMN2HTTRECQL
SCHEMBL8973048 0.79 MAPT (0.50) EPHX2SIGMAR1SMN1; SMN2CES2CES1
SCHEMBL4533824 0.78 HRH3 (0.55) CYP1A2CYP2D6KCNH2
SCHEMBL4481722 0.78 HRH3 (0.58) CYP1A2CYP2D6KCNH2
SCHEMBL6136613 0.78 CYP1A2 (0.50) EPHX2HTTMAPTPOLBCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105121404-A Aryl sulfonamide and sulfamic acid derivatives as RORc modulators HOFFMANN LA ROCHE 2015-12-02 CN disclosed