SCHEMBL28045972

SCHEMBL28045972

Cc1c(C=O)ccc(O)c1N(C)C

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 9/20 0.38
TYR P14679 2/20 0.38
TRIM24 O15164 2/20 0.38
TRIM33 Q9UPN9 2/20 0.38
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
HSP90AA1 P07900 1/20 0.35
IDO1 P14902 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PIM1 P11309 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
KCNJ1 P48048 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1002718 0.77 TRIM24 (0.44) ERN1TYRTRIM24TRIM33KDM4E
SCHEMBL29459676 0.77 TRIM24 (0.44) ERN1TYRTRIM24TRIM33KDM4E
SCHEMBL29459704 0.75 ERN1 (0.50) ERN1TYRTRIM24TRIM33KDM4E
SCHEMBL670303 0.75 ERN1 (0.50) ERN1TYRTRIM24TRIM33KDM4E
SCHEMBL12760732 0.74 ERN1 (0.55) ERN1TYRTRIM24TRIM33ALDH1A1
SCHEMBL3965959 0.73 TRPA1 (0.41) KDM4EALDH1A1KMT2ANPSR1PIM1
SCHEMBL18729174 0.72 ERN1 (0.48) ERN1TYRTRIM24TRIM33KDM4E
SCHEMBL767452 0.71 ERN1 (0.50) ERN1TYRTRIM24TRIM33KDM4E
SCHEMBL30400746 0.71 ERN1 (0.50) ERN1TYRTRIM24TRIM33KDM4E
SCHEMBL5724597 0.71 ERN1 (0.46) ERN1TYRTRIM24TRIM33ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105189485-B It is used as the novel propylene amide derivatives of anti-malarial agents 埃科特莱茵药品有限公司 2017-10-24 CN disclosed
CN-105189485-A Novel acrylamide derivatives as antimalarial agents ACTELION PHARMACEUTICALS LTD 2015-12-23 CN disclosed