SCHEMBL28046090

SCHEMBL28046090

C=CCOC(=O)Nc1cccc(OC(N)=O)c1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
CASP1 P29466 4/20 0.38
KDM4E B2RXH2 3/20 0.37
HSD17B10 Q99714 2/20 0.37
MAPK1 P28482 2/20 0.37
CYP3A4 P08684 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ALDH1A1 P00352 3/20 0.35
TSHR P16473 2/20 0.35
CSNK2A2 P19784 1/20 0.35
CSNK2A1 P68400 1/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
POLB P06746 3/20 0.34
LIG1 P18858 1/20 0.34
HPGD P15428 1/20 0.34
KCNQ3 O43525 1/20 0.33
KCNQ2 O43526 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1127560 0.76 CYP1A2 (0.48) KMT2AMEN1CASP1KDM4EHSD17B10
SCHEMBL27798244 0.75 RXFP1 (0.43) KDM4EALDH1A1NPC1RAB9ANPSR1
SCHEMBL11782094 0.74 KMT2A (0.49) KMT2AMEN1HSD17B10MAPK1CYP3A4
SCHEMBL20049003 0.73 MEN1 (0.44) KMT2AMEN1KDM4EHSD17B10MAPK1
SCHEMBL27834650 0.72 KMT2A (0.51) KMT2AMEN1MAPK1CYP3A4TSHR
SCHEMBL18506525 0.71 MEN1 (0.50) KMT2AMEN1KDM4EHSD17B10MAPK1
SCHEMBL3562718 0.71 MEN1 (0.53) KMT2AMEN1HSD17B10MAPK1ALDH1A1
SCHEMBL5972595 0.71 KMT2A (0.56) KMT2AMEN1CASP1KDM4EHSD17B10
SCHEMBL9271743 0.70 ALDH1A1 (0.67) KMT2AMEN1CASP1KDM4EHSD17B10
SCHEMBL31370710 0.70 KMT2A (0.55) KMT2AMEN1CASP1KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105228983-A The compound regulated for kinases and indication thereof PLEXXIKON INC 2016-01-06 CN disclosed