SCHEMBL28046571

SCHEMBL28046571

CC(=O)Nc1ccc2c(ccn2Cc2ccc(C)cc2)c1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.58
HDAC6 Q9UBN7 2/20 0.58
HDAC3 O15379 1/20 0.58
HDAC1 Q13547 1/20 0.58
HDAC2 Q92769 1/20 0.58
KCNQ3 O43525 2/20 0.56
KCNQ2 O43526 2/20 0.56
KCNQ4 P56696 2/20 0.56
KCNQ5 Q9NR82 2/20 0.56
CHRNA7 P36544 2/20 0.52
KCNH2 Q12809 1/20 0.52
MAOB P27338 1/20 0.52
EPHX2 P34913 7/20 0.51
ALOX5 P09917 2/20 0.49
HDAC11 Q96DB2 1/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
LMNA P02545 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6086484 0.90 KCNQ3 (0.56) HDAC8HDAC6HDAC3HDAC1HDAC2
SCHEMBL28046564 0.89 KCNQ3 (0.55) HDAC8HDAC6HDAC3HDAC1HDAC2
SCHEMBL6085966 0.88 KCNQ3 (0.55) HDAC8HDAC6HDAC3HDAC1HDAC2
SCHEMBL28046562 0.88 HDAC8 (0.64) HDAC8HDAC6HDAC3HDAC1HDAC2
SCHEMBL15601460 0.88 KCNQ3 (0.56) HDAC8HDAC6KCNQ3KCNQ2KCNQ4
SCHEMBL15601447 0.86 KCNQ3 (0.53) HDAC8HDAC6HDAC3HDAC1HDAC2
SCHEMBL15601462 0.86 EPHX2 (0.64) HDAC8HDAC6HDAC3HDAC1HDAC2
SCHEMBL15601409 0.86 KCNQ3 (0.65) HDAC8HDAC6HDAC3HDAC1HDAC2
SCHEMBL15601468 0.85 KCNQ3 (0.53) HDAC8HDAC6KCNQ3KCNQ2KCNQ4
SCHEMBL15601449 0.85 KCNQ3 (0.55) HDAC8HDAC6HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103554008-B 1,3-replacement-5-acetylamino indole ketone compound and the application in antineoplastic thereof TIANJIN UNIVERSITY OF SCIENCE & TECHNOLOGY (CN) 2016-05-04 CN disclosed