SCHEMBL28046993

SCHEMBL28046993

Cc1c(CN2CCN(C(=O)N3CCN(Cc4cc(F)cc([N+](=O)[O-])c4C)CC3C)C(C)C2)cc(F)cc1[N+](=O)[O-]

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.49
RORC P51449 7/20 0.47
ALDH1A1 P00352 3/20 0.43
MAPT P10636 2/20 0.43
MGLL Q99685 1/20 0.39
FAAH O00519 1/20 0.39
LMNA P02545 1/20 0.38
CCR1 P32246 2/20 0.38
THRB P10828 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
KDM4E B2RXH2 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
TACR1 P25103 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18787549 0.93 KCNH2 (0.47) KCNH2RORCALDH1A1MAPTMGLL
SCHEMBL17295599 0.93 KCNH2 (0.47) KCNH2RORCALDH1A1MAPTMGLL
SCHEMBL15778101 0.88 KCNH2 (0.64) KCNH2RORC
SCHEMBL15778102 0.88 KCNH2 (0.64) KCNH2RORC
SCHEMBL15777777 0.87 ALDH1A1 (0.47) KCNH2RORCALDH1A1MAPTLMNA
SCHEMBL17182378 0.87 ALDH1A1 (0.47) KCNH2RORCALDH1A1MAPTLMNA
SCHEMBL19381059 0.86 KCNH2 (0.47) KCNH2RORCALDH1A1MAPTCCR1
SCHEMBL17182361 0.85 KCNH2 (0.46) KCNH2RORCALDH1A1MAPTMGLL
SCHEMBL15778171 0.85 KCNH2 (0.46) KCNH2RORCALDH1A1MAPTMGLL
SCHEMBL18695721 0.85 KCNH2 (0.52) KCNH2RORCALDH1A1MAPTTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105121430-A Modulators of the retinoid-related orphan receptor gamma (ror-gamma) for use in the treatment of autoimmune and inflammatory diseases GLAXO GROUP LTD 2015-12-02 CN disclosed