SCHEMBL28047026

SCHEMBL28047026

CCOC(=O)c1oc2cc(Cl)c(O)cc2c1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.53
RAB9A P51151 2/20 0.53
NPC1 O15118 1/20 0.53
HIF1A Q16665 7/20 0.51
GPR35 Q9HC97 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
USP2 O75604 1/20 0.48
BRAF P15056 1/20 0.47
EIF2AK3 Q9NZJ5 1/20 0.47
KDM4E B2RXH2 3/20 0.47
AHR P35869 1/20 0.47
TSHR P16473 2/20 0.47
PARG Q86W56 2/20 0.46
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
ALOX15 P16050 1/20 0.46
CASP1 P29466 1/20 0.46
CASP7 P55210 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3640665 0.94 MAPT (0.53) MAPTRAB9ANPC1HIF1AGPR35
SCHEMBL10743403 0.88 GPR35 (0.64) MAPTRAB9ANPC1HIF1AGPR35
SCHEMBL28047029 0.84 HIF1A (0.51) MAPTRAB9ANPC1HIF1AL3MBTL1
SCHEMBL3646419 0.81 HIF1A (0.51) MAPTRAB9ANPC1HIF1AL3MBTL1
SCHEMBL24470709 0.81 KMT2A (0.58) MAPTNPC1HIF1AL3MBTL1KDM4E
SCHEMBL29713164 0.81 KMT2A (0.58) MAPTNPC1HIF1AL3MBTL1KDM4E
SCHEMBL11698424 0.80 KDM4E (0.47) MAPTRAB9ANPC1HIF1AL3MBTL1
SCHEMBL3648813 0.79 BRAF (0.44) MAPTRAB9ANPC1HIF1AL3MBTL1
SCHEMBL20893367 0.79 MCL1 (0.67) MAPTRAB9ANPC1HIF1AL3MBTL1
SCHEMBL9378819 0.79 KDM4E (0.69) MAPTRAB9AHIF1AUSP2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105164112-A Amide compound and preparation method, pharmaceutical composition and application thereof SHANGHAI INST MATERIA MEDICA 2015-12-16 CN disclosed