SCHEMBL28048972

SCHEMBL28048972

CC(C)(C)OC(=O)Nc1sc(-c2cc(Br)cc(F)c2F)nc1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LCK P06239 7/20 0.39
AAK1 Q2M2I8 4/20 0.33
BRAF P15056 1/20 0.31
SYK P43405 1/20 0.31
CYP17A1 P05093 1/20 0.31
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28048977 0.88 S1PR3 (0.34) LCKBRAF
SCHEMBL2525712 0.88 AAK1 (0.40) LCKAAK1
SCHEMBL2521268 0.88 LCK (0.37) LCKAAK1BRAFSYK
SCHEMBL2522570 0.83 LCK (0.38) LCKSYK
SCHEMBL28048973 0.82 LCK (0.34) LCKCA1CA2
SCHEMBL2518575 0.81 NPC1 (0.38) LCKSYK
SCHEMBL2518546 0.81 LCK (0.37) LCKAAK1
SCHEMBL2523163 0.81 PIM1 (0.36) LCKBRAFSYKCYP17A1
SCHEMBL2523289 0.81 MAPT (0.39) LCKCYP17A1
SCHEMBL6524464 0.80 ACVR1B (0.40) LCKBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102625807-B 4-Substituted pyridin-3-yl-carboxamide compounds and methods of use HOFFMAN-LA ROCHE LTD. (CH) 2016-03-09 CN disclosed