SCHEMBL28048977

SCHEMBL28048977

CC(C)(C)OC(=O)Nc1sc(-c2cc(Cl)cc(F)c2F)nc1C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 1/20 0.34
LCK P06239 5/20 0.33
BDKRB1 P46663 3/20 0.33
ACVR1B P36896 1/20 0.33
TGFBR1 P36897 1/20 0.33
ACVRL1 P37023 1/20 0.33
BRAF P15056 1/20 0.33
P2RX3 P56373 3/20 0.32
ADORA3 P0DMS8 1/20 0.32
ADORA2B P29275 1/20 0.32
MAPKAPK2 P49137 1/20 0.32
RORC P51449 1/20 0.32
AGPAT2 O15120 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6524464 0.88 ACVR1B (0.40) S1PR3LCKACVR1BTGFBR1ACVRL1
SCHEMBL28048972 0.88 LCK (0.39) LCKBRAF
SCHEMBL2523163 0.83 PIM1 (0.36) LCKBRAF
SCHEMBL2522570 0.83 LCK (0.38) LCK
SCHEMBL14800615 0.82 PIM1 (0.37) LCKBRAF
SCHEMBL2518575 0.81 NPC1 (0.38) LCKADORA3ADORA2B
SCHEMBL2521268 0.81 LCK (0.37) LCKBRAF
SCHEMBL2523289 0.81 MAPT (0.39) LCKRORC
SCHEMBL15573656 0.81 LCK (0.41) LCKBRAF
SCHEMBL2522933 0.79 PIM1 (0.41) LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102625807-B 4-Substituted pyridin-3-yl-carboxamide compounds and methods of use HOFFMAN-LA ROCHE LTD. (CH) 2016-03-09 CN disclosed