SCHEMBL28048979

SCHEMBL28048979

Nc1ccc2[nH]c(C34CC5CC(CC(C5)C3)C4)cc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
LMNA P02545 2/20 0.46
CYP2A6 P11509 1/20 0.45
KEAP1 Q14145 1/20 0.45
MAPT P10636 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
USP2 O75604 1/20 0.39
THRB P10828 1/20 0.39
HRH4 Q9H3N8 1/20 0.38
TSHR P16473 1/20 0.37
KDM4E B2RXH2 2/20 0.36
HPGD P15428 2/20 0.36
HSD17B10 Q99714 1/20 0.36
NPY5R Q15761 1/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
GAA P10253 2/20 0.34
ROCK2 O75116 1/20 0.34
RAB9A P51151 1/20 0.34
ROCK1 Q13464 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11820426 0.79 CNR2 (0.50) ALDH1A1LMNACYP2A6MAPTTDP1
SCHEMBL30435190 0.79 CNR2 (0.50) ALDH1A1LMNACYP2A6MAPTTDP1
SCHEMBL28049107 0.75 KDM4E (0.37) ALDH1A1MAPTTDP1USP2THRB
SCHEMBL1465854 0.72 CYP2A6 (0.53) ALDH1A1CYP2A6KEAP1MAPTTDP1
SCHEMBL24524235 0.70 ALDH1A1 (0.67) ALDH1A1LMNAMAPTTDP1KDM4E
SCHEMBL31289515 0.67 ALDH1A1 (0.51) ALDH1A1LMNAMAPTTDP1USP2
SCHEMBL6019304 0.66 CYP2A6 (0.63) ALDH1A1CYP2A6KEAP1MAPTTDP1
SCHEMBL10172983 0.66 CYP2A6 (0.63) ALDH1A1LMNACYP2A6KEAP1MAPT
SCHEMBL1465598 0.65 CYP2A6 (0.52) ALDH1A1CYP2A6KEAP1MAPTTDP1
SCHEMBL399431 0.64 ALDH1A1 (1.00) ALDH1A1LMNAMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113845461-A 4- (2-adamantane-1H-indol-5-yl) semicarbazide derivative and preparation method and application thereof 浙江师范大学行知学院 2021-12-28 CN claimed
CN-113845461-B 4- (2-adamantane-1H-indol-5-yl) semicarbazide derivative and preparation method and application thereof 浙江师范大学行知学院 2023-06-20 CN disclosed
CN-113845461-A 4- (2-adamantane-1H-indol-5-yl) semicarbazide derivative and preparation method and application thereof 浙江师范大学行知学院 2021-12-28 CN disclosed
CN-105348168-A 1-(2-(adamantane-1-yl)-1H-indole-5-yl)-3-substituted urea derivative, preparation and use thereof UNIV XIAMEN 2016-02-24 CN disclosed