SCHEMBL28049564

SCHEMBL28049564

Nc1cc(N)nc(C2CCNC2)n1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 3/20 0.45
HTR3A P46098 1/20 0.39
MPO P05164 1/20 0.38
CHEK1 O14757 1/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
CCNA1 P78396 1/20 0.36
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
PARP1 P09874 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2034798 0.89 CHEK1 (0.47) HRH4CHEK1CCNA2CDK2CCNA1
SCHEMBL2403564 0.88 HRH4 (0.50) HRH4HTR2C
SCHEMBL28063327 0.79 HRH3 (0.42) HRH4HTR3ACHEK1CCNA2CDK2
SCHEMBL2637316 0.77 TLR9 (0.39) HTR3AMPOHTR2AHTR2C
SCHEMBL20577260 0.77 TLR9 (0.39) HTR3AMPOHTR2AHTR2C
SCHEMBL16789827 0.77 PDE10A (0.42) HRH4
SCHEMBL14240499 0.77 HRH4 (0.44) HRH4HTR2C
SCHEMBL28383379 0.75 HRH4 (0.33) HRH4
SCHEMBL28460425 0.73 HRH4 (0.40) HRH4HTR3AMPOCHEK1CCNA2
SCHEMBL2176046 0.71 BACE1 (0.44) HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105367503-A HETEROARYL COMPOUNDS AND USES THEREOF AVILA THERAPEUTICS INC 2016-03-02 CN disclosed
CN-101902911-B Heteroaryl compounds and uses thereof AVILA THERAPEUTICS, INC. (US) 2015-12-16 CN disclosed