SCHEMBL28049640

SCHEMBL28049640

CC#Cc1cc(C(=O)O)ccc1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.46
RXRA P19793 1/20 0.43
RXRB P28702 1/20 0.43
MYC P01106 1/20 0.42
ESR1 P03372 1/20 0.42
ALOX15 P16050 1/20 0.42
PTPN7 P35236 1/20 0.42
HSD17B10 Q99714 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
TPMT P51580 2/20 0.42
ALDH1A1 P00352 2/20 0.42
GRM1 Q13255 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
KMT2A Q03164 1/20 0.41
GAA P10253 2/20 0.41
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1712869 0.81 MYC (0.45) TSHRRXRARXRBMYCHSD17B10
SCHEMBL3420562 0.81 TSHR (0.42) TSHRMYCESR1ALOX15PTPN7
SCHEMBL14616920 0.81 HAO1 (0.50) TSHR
SCHEMBL3959215 0.79 ALDH1A1 (0.51) TSHRMYCESR1ALOX15PTPN7
SCHEMBL31186416 0.79 ALDH1A1 (0.51) TSHRMYCESR1ALOX15PTPN7
SCHEMBL9609642 0.79 TSHR (0.47) TSHRRXRARXRBMYCESR1
SCHEMBL24528448 0.77 TDP1 (0.42) TSHRMYCESR1ALOX15PTPN7
SCHEMBL9609638 0.77 TSHR (0.40) TSHRRXRAMYCESR1ALOX15
SCHEMBL4062149 0.76 CSF1R (0.46) TSHR
SCHEMBL566400 0.75 ALDH1A1 (0.42) TSHRRXRAALDH1A1TDP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103965195-B Compound and application thereof for discoidin domain receptor micromolecular inhibitor 中国科学院广州生物医药与健康研究院 2016-09-28 CN disclosed
CN-103214480-B Pyrazolopyridine alkynes benzene-like compounds and medicinal compositions thereof and application GUANGZHOU INSTITUTES OF BIOMEDICINE AND HEALTH, CHINESE ACADEMY OF SCIENCES (CN) 2015-12-16 CN disclosed
CN-103965195-A Compound used for discoidin domain receptor micro-molecule inhibitor, and its application GUANGZHOU INST BIOMED & HEALTH 2014-08-06 CN disclosed