SCHEMBL28050302

SCHEMBL28050302

COc1ccc(CN2CC(OC(C)=O)CCC2=O)cc1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
MMP1 P03956 1/20 0.47
MMP13 P45452 1/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2C19 P33261 2/20 0.47
KMT2A Q03164 3/20 0.46
GAA P10253 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
GRM2 Q14416 1/20 0.44
POLB P06746 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28006519 0.88 ALDH1A1 (0.54) ALDH1A1L3MBTL1MMP1MMP13CYP3A4
SCHEMBL27956316 0.83 BTK (0.49) ALDH1A1KMT2APOLBSMN1; SMN2
SCHEMBL17062184 0.81 GAA (0.50) ALDH1A1L3MBTL1MMP1MMP13CYP3A4
SCHEMBL16759341 0.81 GAA (0.50) ALDH1A1L3MBTL1MMP1MMP13CYP3A4
SCHEMBL3488361 0.80 SMN1; SMN2 (0.55) ALDH1A1L3MBTL1CYP3A4CYP2C19KMT2A
SCHEMBL16485924 0.79 KMT2A (0.53) ALDH1A1L3MBTL1CYP3A4CYP2C19KMT2A
SCHEMBL3488893 0.79 KMT2A (0.56) ALDH1A1L3MBTL1CYP3A4CYP2C19KMT2A
SCHEMBL22488324 0.79 KDM4E (0.53) KMT2A
SCHEMBL22468572 0.79 KDM4E (0.53) KMT2A
SCHEMBL16485861 0.78 GAA (0.50) ALDH1A1L3MBTL1MMP1MMP13CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105408330-A Novel aza-oxo-indoles for the treatment and prophylaxis of respiratory syncytial virus infection HOFFMANN LA ROCHE 2016-03-16 CN disclosed