SCHEMBL28050840

SCHEMBL28050840

Cc1cnc(C)c(-n2ccnn2)c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 14/20 0.46
EGLN2 Q96KS0 2/20 0.42
HCRTR2 O43614 2/20 0.36
HCRTR1 O43613 1/20 0.35
KEAP1 Q14145 1/20 0.34
CYP19A1 P11511 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CHRNB2 P17787 1/20 0.33
CYP2B6 P20813 1/20 0.33
MAOA P21397 1/20 0.33
CYP2C19 P33261 1/20 0.33
CHRNA4 P43681 1/20 0.33
HTR3A P46098 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14909053 0.83 NOTUM (0.42) NOTUMEGLN2KEAP1CYP19A1CYP1A2
SCHEMBL16039381 0.79 HCRTR2 (0.43) NOTUMEGLN2HCRTR2HCRTR1
SCHEMBL16031459 0.79 NOTUM (0.40) NOTUMEGLN2HCRTR2HCRTR1CYP19A1
SCHEMBL20912232 0.75 ALDH1A1 (0.47) NOTUM
SCHEMBL16113420 0.73 NOTUM (0.47) NOTUMEGLN2HCRTR2HCRTR1KEAP1
SCHEMBL22642750 0.72 NOTUM (0.50) NOTUMEGLN2HCRTR2HCRTR1CYP1A2
SCHEMBL28361867 0.70 NOTUM (0.44) NOTUMEGLN2HCRTR2HCRTR1KEAP1
SCHEMBL21030734 0.70 NOTUM (0.42) NOTUMEGLN2HCRTR2HCRTR1CYP19A1
SCHEMBL5612789 0.69 NOTUM (0.56) NOTUMEGLN2KEAP1CYP19A1
SCHEMBL30046228 0.69 NOTUM (0.56) NOTUMEGLN2KEAP1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105209468-A Substituted 7-azabicycles and their use as orexin receptor modulators JANSSEN PHARMACEUTICA NV 2015-12-30 CN disclosed