SCHEMBL28051001

SCHEMBL28051001

COc1ccc2cc(Cc3ccc(F)cc3)ccc2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 5/20 0.42
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
TXNRD1 Q16881 1/20 0.40
PDE10A Q9Y233 4/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
STAT3 P40763 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
HTR1A P08908 1/20 0.38
HTR3A P46098 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38
TLR2 O60603 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28269737 0.87 MAOB (0.40) MTNR1AMTNR1BPDE10AMAPTSMN1; SMN2
SCHEMBL27987661 0.85 TEC (0.45) MTNR1AMTNR1BTXNRD1PDE10ALMNA
SCHEMBL30081479 0.82 BACE1 (0.53) MTNR1AMTNR1BPDE10AMAPTBACE1
SCHEMBL19808389 0.79 CYP1A2 (0.46) MTNR1AMTNR1BPDE10ALMNAMAPT
SCHEMBL28269735 0.78 PDE10A (0.41) MTNR1AMTNR1BPDE10ASMN1; SMN2HDAC3
SCHEMBL21458325 0.78 MTNR1A (0.47) MTNR1AMTNR1BPDE10AAPPHDAC3
SCHEMBL31731406 0.78 MTNR1A (0.47) MTNR1AMTNR1BPDE10AAPPHDAC3
SCHEMBL28271357 0.75 PDE10A (0.45) PDE10A
SCHEMBL11830895 0.75 MTNR1A (0.45) MTNR1AMTNR1BPDE10ALMNAPOLB
SCHEMBL11832008 0.75 MTNR1A (0.51) MTNR1AMTNR1BPDE10ALMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105829294-A METHYLENE LINKED QUINOLINYL MODULATORS OF ROR-GAMMA-T 詹森药业有限公司 2016-08-03 CN disclosed
CN-105636952-A Secondary alcohol quinolinyl modulators of roryt JANSSEN PHARMACEUTICA NV 2016-06-01 CN disclosed
CN-105209453-A Methylene linked quinolinyl modulators of ROR-gamma-T JANSSEN PHARMACEUTICA NV 2015-12-30 CN disclosed