SCHEMBL28051301

SCHEMBL28051301

NCc1ccc(C(N)=O)c(-c2nccs2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 1/20 0.53
CHEK2 O96017 1/20 0.41
ROCK1 Q13464 1/20 0.37
HPGD P15428 1/20 0.37
CYP2A6 P11509 1/20 0.36
ADRB2 P07550 1/20 0.36
THRA P10827 1/20 0.36
THRB P10828 1/20 0.36
TYK2 P29597 1/20 0.36
PDPK1 O15530 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
MYC P01106 1/20 0.35
FFAR1 O14842 1/20 0.35
MAPK8 P45983 3/20 0.34
PLA2G2A P14555 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27664694 0.81 CHEK2 (0.53) CHEK2TYK2MEN1ALDH1A1MAPT
SCHEMBL995828 0.76 CSNK1A1 (0.50) CHEK2HPGDTYK2PDPK1MEN1
SCHEMBL30517722 0.76 CSNK1A1 (0.50) CHEK2HPGDTYK2PDPK1MEN1
SCHEMBL30576812 0.75 KDM4E (0.47) HPGDALDH1A1MAPT
Hydrochloric Acid SCHEMBL30810223 0.75 CSNK1A1 (0.49) CHEK2HPGDTYK2PDPK1MEN1
SCHEMBL5698784 0.75 KDM4E (0.40) CHEK2HPGDTYK2PDPK1MEN1
SCHEMBL30576798 0.75 KDR (0.41) MAPK8
SCHEMBL28843050 0.74 PLA2G2A (0.44) LOXL2CHEK2PDPK1PTGDR2FFAR1
SCHEMBL918767 0.74 CSNK1A1 (0.48) CHEK2TYK2PDPK1MEN1ALDH1A1
SCHEMBL27986525 0.74 CHEK2 (0.45) LOXL2CHEK2ROCK1CYP2A6THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102812006-B Novel antimalaria reagent MMV MEDICINES FOR MALARIA VENTURE (CH) 2016-01-20 CN disclosed