SCHEMBL28051628

SCHEMBL28051628

NC(=O)c1ccc(-c2ccc(C3CCNCC3)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.51
PARP1 P09874 4/20 0.51
PARP2 Q9UGN5 1/20 0.51
P2RY14 Q15391 7/20 0.48
SIGMAR1 Q99720 2/20 0.47
SLC18A3 Q16572 1/20 0.47
HTR2C P28335 2/20 0.45
QDPR P09417 1/20 0.45
DGAT1 O75907 1/20 0.44
PDE2A O00408 1/20 0.44
PDE5A O76074 1/20 0.44
EGFR P00533 1/20 0.44
INSR P06213 1/20 0.44
HTR1A P08908 1/20 0.44
ADRA2A P08913 1/20 0.44
ADRB3 P13945 1/20 0.44
ADRA2B P18089 1/20 0.44
ADRA2C P18825 1/20 0.44
DRD1 P21728 1/20 0.44
DRD5 P21918 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28051650 0.98 PARP1 (0.50) CYP2C9PARP1PARP2P2RY14SIGMAR1
SCHEMBL1758181 0.95 CYP2C9 (0.55) CYP2C9PARP1PARP2SIGMAR1SLC18A3
Hydrochloric Acid SCHEMBL3630728 0.93 CYP2C9 (0.54) CYP2C9PARP1PARP2SIGMAR1SLC18A3
Hydrochloric Acid SCHEMBL28051652 0.89 PARP1 (0.52) PARP1PARP2
SCHEMBL12607512 0.85 HTR2C (0.48) PARP1PARP2P2RY14SIGMAR1SLC18A3
SCHEMBL12505084 0.85 HTR3A (0.56) PARP1
Trifluoroacetic Acid SCHEMBL6703422 0.84 HTR2C (0.51) CYP2C9PARP1PARP2P2RY14SIGMAR1
Hydrochloric Acid SCHEMBL1790636 0.84 HTR2C (0.49) PARP1PARP2P2RY14SIGMAR1SLC18A3
Hydrochloric Acid SCHEMBL4200472 0.83 HTR3A (0.54) PARP1
Hydrochloric Acid SCHEMBL4200477 0.83 HTR3A (0.54) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105254623-A SUBSTITUTED BENZAMIDES HOFFMANN LA ROCHE 2016-01-20 CN claimed
CN-105254623-A SUBSTITUTED BENZAMIDES HOFFMANN LA ROCHE 2016-01-20 CN disclosed