SCHEMBL28053995

SCHEMBL28053995

C=CC(=O)Nc1cc(Nc2ncc(Cl)c(Nc3ccc(N4CCOCC4)cc3OC)n2)c(OC)cc1N(C)CCN(C)C

nearest known ligand 0.68

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EGFR P00533 17/20 0.68
ALK Q9UM73 6/20 0.67
EML4 Q9HC35 3/20 0.67
INSR P06213 3/20 0.65
ERBB2 P04626 1/20 0.65
ROS1 P08922 1/20 0.65
FER P16591 1/20 0.65
LTK P29376 1/20 0.65
BLK P51451 1/20 0.65
PTK2 Q05397 1/20 0.65
BTK Q06187 1/20 0.65
TNK2 Q07912 1/20 0.65
ERBB4 Q15303 1/20 0.65
SLK Q9H2G2 1/20 0.65
CYP3A4 P08684 1/20 0.61
CYP2C9 P11712 1/20 0.61
CYP2C19 P33261 1/20 0.61
KCNH2 Q12809 1/20 0.61
MAPK3 P27361 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17059222 0.89 EGFR (0.73) EGFRALKEML4INSRKCNH2
SCHEMBL17059193 0.86 EGFR (0.69) EGFRALKEML4INSRKCNH2
SCHEMBL28053871 0.86 EGFR (0.75) EGFRALKINSRERBB2ROS1
Hydrochloric Acid SCHEMBL28053993 0.85 EGFR (0.74) EGFRALKINSRERBB2ROS1
SCHEMBL17059288 0.85 EGFR (0.74) EGFR
SCHEMBL28053863 0.84 ALK (0.66) EGFRALKINSRERBB2ROS1
SCHEMBL28053865 0.84 EGFR (0.83) EGFRALKINSRERBB2ROS1
SCHEMBL17059269 0.83 EGFR (0.72) EGFRALKEML4
Hydrochloric Acid SCHEMBL28053870 0.83 EGFR (0.82) EGFRALKINSRERBB2ROS1
SCHEMBL17059323 0.83 EGFR (0.69) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105384694-B Substituted aminopyrimidine derivative and preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2020-09-04 CN disclosed
CN-105384694-A Substituted aminopyrimidine derivative, preparation method therefor and pharmaceutical application thereof SICHUAN HAISCO PHARMACEUTICAL CO LTD 2016-03-09 CN disclosed