SCHEMBL28053865

SCHEMBL28053865

C=CC(=O)Nc1ccc(OC)c(Nc2ncc(Cl)c(Nc3ccc(N4CCOCC4)cc3OC)n2)c1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.83
INSR P06213 2/20 0.72
ALK Q9UM73 2/20 0.72
MAPK8 P45983 2/20 0.68
MAPK9 P45984 2/20 0.68
MAPK10 P53779 2/20 0.68
LRRK2 Q5S007 2/20 0.67
CDC7 O00311 1/20 0.67
PLK4 O00444 1/20 0.67
CHEK1 O14757 1/20 0.67
AURKA O14965 1/20 0.67
DCLK1 O15075 1/20 0.67
PDPK1 O15530 1/20 0.67
DAPK3 O43293 1/20 0.67
DYRK3 O43781 1/20 0.67
JAK2 O60674 1/20 0.67
PRKD3 O94806 1/20 0.67
PAK4 O96013 1/20 0.67
CHEK2 O96017 1/20 0.67
ERBB2 P04626 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28053870 0.99 EGFR (0.82) EGFRINSRALKMAPK8MAPK9
SCHEMBL28445838 0.92 EGFR (0.80) EGFRINSRALKMAPK8MAPK9
SCHEMBL28053891 0.92 JAK3 (0.77) EGFRALKPLK4JAK2FLT3
SCHEMBL2722635 0.91 EGFR (1.00) EGFRINSRALKPLK4JAK2
SCHEMBL28579656 0.90 EGFR (0.83) EGFRALKMAPK3
SCHEMBL28589279 0.89 ALK (0.71) EGFRINSRALKAURKAIGF1R
SCHEMBL28053991 0.89 JAK3 (0.73) EGFRALKPLK4JAK2FLT3
SCHEMBL28053871 0.89 EGFR (0.75) EGFRINSRALKMAPK8MAPK9
Hydrochloric Acid SCHEMBL28053993 0.88 EGFR (0.74) EGFRINSRALKMAPK8MAPK9
SCHEMBL28447722 0.87 EGFR (0.78) EGFRALKJAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105384694-B Substituted aminopyrimidine derivative and preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2020-09-04 CN disclosed
CN-105384694-A Substituted aminopyrimidine derivative, preparation method therefor and pharmaceutical application thereof SICHUAN HAISCO PHARMACEUTICAL CO LTD 2016-03-09 CN disclosed