SCHEMBL28055284

SCHEMBL28055284

CC(C)(C(=O)OC(=O)C(F)(F)F)n1cc(-c2ccnc3[nH]ccc23)cn1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AURKA O14965 4/20 0.54
AURKB Q96GD4 4/20 0.54
INCENP Q9NQS7 2/20 0.54
TPX2 Q9ULW0 2/20 0.54
GRM4 Q14833 1/20 0.50
JAK1 P23458 3/20 0.48
JAK2 O60674 8/20 0.46
NUDT1 P36639 1/20 0.44
CIT O14578 2/20 0.43
IKBKB O14920 1/20 0.43
CHUK O15111 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL5134407 0.86 AURKB (0.57) AURKAAURKBINCENPTPX2GRM4
Trifluoroacetic Acid SCHEMBL100051 0.85 AURKA (0.49) AURKAAURKBINCENPTPX2GRM4
SCHEMBL98741 0.84 AURKA (0.55) AURKAAURKBINCENPTPX2GRM4
SCHEMBL13774666 0.84 AURKB (0.62) AURKAAURKBINCENPTPX2GRM4
SCHEMBL100576 0.84 AURKB (0.62) AURKAAURKBINCENPTPX2GRM4
SCHEMBL15399202 0.84 JAK2 (0.63) JAK1JAK2
SCHEMBL99617 0.84 AURKA (0.49) AURKAAURKBINCENPTPX2GRM4
SCHEMBL99011 0.83 AURKB (0.60) AURKAAURKBINCENPTPX2GRM4
SCHEMBL4094038 0.82 JAK2 (0.51) AURKAAURKBINCENPTPX2GRM4
SCHEMBL14845593 0.82 AURKB (0.59) AURKAAURKBINCENPTPX2GRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103214484-B Pyrrolo-[2,3-b] pyridine replaced as the heteroaryl of Janus inhibitors of kinases and pyrrolo-[2,3-b] pyrimidine 因塞特控股公司 2016-07-06 CN disclosed