SCHEMBL28055302

SCHEMBL28055302

CC(C)(C)OC(=O)c1cc(N)cc2nc3ccccc3cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.41
GAA P10253 5/20 0.40
KMT2A Q03164 4/20 0.40
MEN1 O00255 3/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
IKBKB O14920 1/20 0.40
KDM4E B2RXH2 7/20 0.40
ALDH1A1 P00352 6/20 0.40
GLA P06280 5/20 0.40
HPGD P15428 5/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
PTBP1 P26599 1/20 0.40
RCE1 Q9Y256 1/20 0.40
ABCG2 Q9UNQ0 2/20 0.40
MAPT P10636 3/20 0.39
HIF1A Q16665 2/20 0.39
THRB P10828 1/20 0.39
ABCB1 P08183 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23632474 0.86 MEN1 (0.44) GAAKMT2AMEN1NPC1RAB9A
SCHEMBL28231808 0.86 MEN1 (0.41) GAAKMT2AMEN1NPC1RAB9A
SCHEMBL28721102 0.85 IKBKB (0.42) GAAKMT2AMEN1NPC1RAB9A
SCHEMBL28230815 0.84 KMT2A (0.47) GAAKMT2AMEN1NPC1RAB9A
SCHEMBL29505627 0.84 KMT2A (0.42) GAAKMT2AMEN1NPC1RAB9A
SCHEMBL29209989 0.84 KMT2A (0.40) GAAKMT2AMEN1NPC1RAB9A
SCHEMBL28720824 0.84 KMT2A (0.42) GAAKMT2AMEN1NPC1RAB9A
SCHEMBL28723805 0.83 KMT2A (0.38) GAAKMT2AMEN1NPC1RAB9A
SCHEMBL28718245 0.81 MEN1 (0.40) GAAKMT2AMEN1NPC1RAB9A
SCHEMBL28231761 0.78 KMT2A (0.44) GAAKMT2AMEN1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111269217-B Pyrimidinamine compound, preparation method and application thereof 苏州信诺维医药科技有限公司 2021-01-08 CN disclosed
CN-111269217-A Pyrimidinamine compound, preparation method and application thereof 苏州信诺维医药科技有限公司 2020-06-12 CN disclosed
CN-110540538-A Inhibitors of influenza virus replication VERTEX PHARMA 2019-12-06 CN disclosed
CN-105294655-A CDK small-molecule inhibitor compounds and application therefore GUANGDONG HEC PHARMACEUTICAL 2016-02-03 CN disclosed