SCHEMBL28055482

SCHEMBL28055482

O=C(O)C#Cc1cccc(Br)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.41
FFAR1 O14842 5/20 0.40
NPSR1 Q6W5P4 3/20 0.40
ALDH1A1 P00352 3/20 0.40
HSP90AA1 P07900 2/20 0.40
MAPT P10636 2/20 0.40
HTT P42858 2/20 0.40
S1PR2 O95136 1/20 0.40
OPRK1 P41145 1/20 0.40
GRM5 P41594 1/20 0.40
HSD17B3 P37058 1/20 0.38
PTPN11 Q06124 1/20 0.38
GFER P55789 1/20 0.37
TP53 P04637 1/20 0.37
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
MITF O75030 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
VCP P55072 1/20 0.36
HNF4A P41235 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL481016 0.79 NPC1 (0.40) PARP1NPSR1ALDH1A1MAPTGRM5
SCHEMBL29779956 0.79 GRM5 (0.53) PARP1ALDH1A1GRM5
SCHEMBL1375869 0.79 GRM5 (0.53) PARP1ALDH1A1GRM5
SCHEMBL27627934 0.78 FFAR1 (0.53) FFAR1NPSR1ALDH1A1HSP90AA1MAPT
SCHEMBL8000068 0.77 APP (0.57) ALDH1A1MAPTGRM5PTPN11TP53
SCHEMBL29825848 0.77 APP (0.57) ALDH1A1MAPTGRM5PTPN11TP53
SCHEMBL3155146 0.77 FFAR1 (0.54) FFAR1ALDH1A1MAPTHTTGRM5
SCHEMBL2235491 0.77 FFAR1 (0.54) FFAR1NPSR1ALDH1A1HSP90AA1MAPT
SCHEMBL5380220 0.77 FFAR1 (0.54) FFAR1NPSR1GRM5VCP
SCHEMBL670363 0.77 CYP2C9 (0.49) PARP1MAPTHTTGRM5PTPN11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116675599-A Novel method for synthesizing phenylpropionic acid 大连理工大学 2023-09-01 CN disclosed
CN-107353194-B Preparation method of propiolic acid compound 大连理工大学 2020-04-14 CN disclosed
CN-105481806-A Synthetic method and application of five-membered ring compound containing sulfone group UNIV SOUTH CHINA TECH 2016-04-13 CN disclosed