SCHEMBL1375869

SCHEMBL1375869

Brc1cccc(C#Cc2cccc(Br)c2)c1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 4/20 0.53
ALDH1A1 P00352 3/20 0.46
MAPK1 P28482 1/20 0.46
APP P05067 1/20 0.43
TDP1 Q9NUW8 1/20 0.38
C1S P09871 1/20 0.38
PARP1 P09874 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
IDO1 P14902 1/20 0.37
AGXT P21549 1/20 0.37
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29779956 1.00 GRM5 (0.53) GRM5ALDH1A1MAPK1APPTDP1
SCHEMBL29825848 0.93 APP (0.57) GRM5ALDH1A1MAPK1APPTDP1
SCHEMBL8000068 0.93 APP (0.57) GRM5ALDH1A1MAPK1APPTDP1
SCHEMBL29868615 0.90 GRM5 (0.46) GRM5ALDH1A1MAPK1APPTDP1
SCHEMBL29288691 0.89 GRM5 (0.46) GRM5ALDH1A1MAPK1APPTDP1
SCHEMBL22202978 0.87 GRM5 (0.45) GRM5ALDH1A1MAPK1TDP1C1S
SCHEMBL4528675 0.87 CA12 (0.50) GRM5ALDH1A1MAPK1TDP1CA12
SCHEMBL10035460 0.87 ALDH1A1 (0.64) GRM5ALDH1A1MAPK1CA12CA1
SCHEMBL14275435 0.87 GRM5 (0.45) GRM5ALDH1A1MAPK1APPC1S
SCHEMBL22203008 0.85 GRM5 (0.44) GRM5ALDH1A1MAPK1TDP1C1S

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117924191-A Polysubstituted olefin derivative and preparation method and application thereof 杭州师范大学 2024-04-26 CN disclosed
CN-108484499-B Method for preparing polysubstituted isoquinoline derivative from hydroxylamine and alkyne 清华大学 2020-06-19 CN disclosed
CN-109897039-A A method of preparing pyrrolo- [3,2,1-ij] quinolinone compounds 中国科学院化学研究所 2019-06-18 CN disclosed
CN-109776546-A A method of preparing indoles and pyrroles's ketone compound 中国科学院化学研究所 2019-05-21 CN disclosed
CN-108484499-A The method that multi-substituted isoquinoline derivative is prepared by azanol and alkynes 清华大学 2018-09-04 CN disclosed
US-9493494-B2 Phosphinine oxide derivative and preparation method thereof KNU-INDUSTRY COOPERATION FOUNDATION (KR) 2016-11-15 US disclosed
US-20150344506-A1 NOVEL PHOSPHININE OXIDE DERIVATIVE AND PREPARATION METHOD THEREOF KNU-INDUSTRY COOPERATION FOUNDATION (KR) 2015-12-03 US disclosed
US-8530607-B2 Aromatic ether and alkynyl containing phthalonitriles THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY OF THE NAVY (US) 2013-09-10 US disclosed
US-20110288254-A1 AROMATIC ETHER AND ALKYNYL CONTAINING PHTHALONITRILES THE GOVERNMENT OF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE NAVY (US) 2011-11-24 US disclosed
US-8039576-B2 Aromatic ether and alkynyl containing phthalonitriles THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE NAVY (US) 2011-10-18 US disclosed
US-7615300-B2 Development of novel proton-conductive polymers for proton exchange membrane fuel cell (PEMFC) technology The Board of Regents University and Community College System of Nevada on Behalf of the University of Nevada (US) 2009-11-10 US disclosed
US-7615300-B2 Development of novel proton-conductive polymers for proton exchange membrane fuel cell (PEMFC) technology The Board of Regents University and Community College System of Nevada on Behalf of the University of Nevada (US) 2009-11-10 US disclosed
US-20090069484-A1 AROMATIC ETHER AND ALKYNYL CONTAINING PHTHALONITRILES THE GOVERNMENT OF THE US, AS REPRESENTED BY THE SECRETARY OF THE NAVY (US) 2009-03-12 US disclosed
US-20070048579-A1 Development of novel proton-conductive polymers for proton exchange membrane fuel cell (PEMFC) technology Board of Regents University and Community College System of Nevada 2007-03-01 US disclosed
US-20070048579-A1 Development of novel proton-conductive polymers for proton exchange membrane fuel cell (PEMFC) technology Board of Regents University and Community College System of Nevada 2007-03-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150344506-A1 NOVEL PHOSPHININE OXIDE DERIVATIVE AND PREPARATION METHOD THEREOF PHOSPHO1, PPIP5K2, ITPA GRM5 732/4885ALDH1A1 3382/4885MAPK1 1506/4885
US-20110288254-A1 AROMATIC ETHER AND ALKYNYL CONTAINING PHTHALONITRILES PNN, BECN1, ACIN1 GRM5 4033/4885ALDH1A1 1956/4885MAPK1 1006/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.