SCHEMBL28055704

SCHEMBL28055704

CC(=O)Nc1ccccc1NCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPRF P10586 1/20 0.56
PTPN2 P17706 1/20 0.56
PTPN1 P18031 1/20 0.56
PTPN11 Q06124 1/20 0.56
MEN1 O00255 6/20 0.53
KMT2A Q03164 6/20 0.53
MAPT P10636 6/20 0.53
GAA P10253 2/20 0.53
CRHBP P24387 2/20 0.52
CRHR2 Q13324 2/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
SMN1; SMN2 Q16637 3/20 0.51
L3MBTL1 Q9Y468 2/20 0.51
HTT P42858 1/20 0.51
CYP19A1 P11511 1/20 0.51
LMNA P02545 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6097282 0.81 CYP19A1 (0.51) MEN1KMT2AMAPTSMN1; SMN2L3MBTL1
SCHEMBL29048560 0.80 MAPT (0.63) PTPRFPTPN2PTPN1PTPN11MEN1
SCHEMBL6170460 0.78 FLT1 (0.47) MEN1KMT2AMAPTGAACRHBP
SCHEMBL18610468 0.77 PTPRF (0.62) PTPRFPTPN2PTPN1PTPN11MEN1
SCHEMBL1804701 0.76 NPC1 (0.58) PTPRFPTPN2PTPN1PTPN11MEN1
SCHEMBL17141871 0.74 PTPRF (0.59) PTPRFPTPN2PTPN1PTPN11MEN1
SCHEMBL4442994 0.74 CCR8 (0.49) CYP19A1LMNA
Acetanilide SCHEMBL27366940 0.72 KMT2A (0.69) MEN1KMT2AMAPTGAACYP1A2
SCHEMBL627885 0.72 PTPRF (1.00) PTPRFPTPN2PTPN1PTPN11MEN1
SCHEMBL1888641 0.72 ABCG2 (0.65) MEN1KMT2AMAPTGAACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105399733-A Novel quinazoline derivative LU1504 and preparing method and application thereof NANJING GENERAL HOSPITAL NANJING MILITARY AREA COMMAND PLA 2016-03-16 CN claimed
CN-105399689-A Novel quinazoline derivative LU1503 and preparing method and application thereof NANJING GENERAL HOSPITAL NANJING MILITARY AREA COMMAND PLA 2016-03-16 CN claimed
CN-105399733-A Novel quinazoline derivative LU1504 and preparing method and application thereof NANJING GENERAL HOSPITAL NANJING MILITARY AREA COMMAND PLA 2016-03-16 CN disclosed
CN-105399689-A Novel quinazoline derivative LU1503 and preparing method and application thereof NANJING GENERAL HOSPITAL NANJING MILITARY AREA COMMAND PLA 2016-03-16 CN disclosed