SCHEMBL28055856

SCHEMBL28055856

NCc1ccccc1-c1ccc(C(=O)Cl)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.58
F10 P00742 3/20 0.46
CYP2C19 P33261 1/20 0.46
KMT2A Q03164 1/20 0.42
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
FOLH1 Q04609 2/20 0.41
HSD17B3 P37058 1/20 0.39
PNMT P11086 1/20 0.38
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
GCG P01275 1/20 0.36
BCL2 P10415 2/20 0.36
BAK1 Q16611 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PTGER1 P34995 1/20 0.35
PTGER4 P35408 1/20 0.35
PTGER3 P43115 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6643039 0.84 PPARA (0.47) CYP2C19KMT2AALDH1A1MAPTL3MBTL1
SCHEMBL7919905 0.84 DPP4 (0.66) DPP4F10CYP2C19KMT2AFOLH1
SCHEMBL30876050 0.81 ALDH1A1 (0.43) KMT2AALDH1A1MAPTL3MBTL1SMN1; SMN2
Bicarbonate SCHEMBL27817695 0.80 DPP4 (0.83) DPP4CYP2C19KMT2AALDH1A1FOLH1
SCHEMBL28154263 0.76 DPP4 (0.47) DPP4F10CYP2C19MAPTHSD17B3
SCHEMBL30466810 0.76 DPP4 (0.69) DPP4F10CYP2C19HSD17B3PNMT
SCHEMBL12524048 0.76 DPP4 (0.69) DPP4CYP2C19KMT2APNMTNOS3
SCHEMBL1134842 0.76 DPP4 (0.69) DPP4F10CYP2C19HSD17B3PNMT
Hydrochloric Acid SCHEMBL7920197 0.75 CYP1A2 (0.51) DPP4CYP2C19KMT2AALDH1A1MAPT
SCHEMBL9146754 0.75 KMT2A (0.46) CYP2C19KMT2AMAPTL3MBTL1FOLH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106029057-A Oral formulations of pyrrolidine derivatives 奥布赛瓦股份公司 2016-10-12 CN disclosed
CN-105531259-A Pyrrolidine derivatives as oxytocin/vasopressin V1a receptor antagonists ObsEva SA 2016-04-27 CN disclosed