SCHEMBL28055971

SCHEMBL28055971

CC(C)(C)C(=O)ON1CCC[C@@H](NC(=O)c2nccs2)C1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TNKS O95271 1/20 0.38
HPGD P15428 1/20 0.37
ALDH1A1 P00352 1/20 0.36
MEN1 O00255 1/20 0.36
TSHR P16473 1/20 0.36
KMT2A Q03164 1/20 0.36
ADORA3 P0DMS8 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA2B P29275 1/20 0.35
USP30 Q70CQ3 3/20 0.35
PBK Q96KB5 1/20 0.35
RBBP9 O75884 1/20 0.35
BTK Q06187 3/20 0.33
HDAC4 P56524 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
GAA P10253 1/20 0.33
JAK3 P52333 1/20 0.33
MGLL Q99685 1/20 0.33
PARP1 P09874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27964022 0.81 RBBP9 (0.41) HPGDALDH1A1MEN1KMT2ARBBP9
SCHEMBL16334091 0.81 USP30 (0.55) ADORA3ADORA2AADORA2BUSP30PBK
SCHEMBL16337990 0.81 USP30 (0.55) ADORA3ADORA2AADORA2BUSP30PBK
SCHEMBL16334556 0.76 TNKS (0.42) TNKSHPGDALDH1A1MEN1TSHR
SCHEMBL28975852 0.75 ALDH1A1 (0.43) HPGDALDH1A1MEN1KMT2ARBBP9
SCHEMBL12181482 0.75 MEN1 (0.54) TNKSHPGDALDH1A1MEN1TSHR
SCHEMBL5738394 0.73 TSHR (0.60) TNKSHPGDALDH1A1MEN1TSHR
SCHEMBL27759531 0.73 USP30 (0.49) ALDH1A1MEN1KMT2AUSP30HDAC4
SCHEMBL28290681 0.72 DRD4 (0.40) ALDH1A1
SCHEMBL27723938 0.72 CA1 (0.37) ALDH1A1USP30BTKGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105530932-B Primary formamide as BTK inhibitor 艾伯维公司 2019-09-27 CN disclosed
CN-105530932-A Primary carboxamides as BIK inhibitors ABBVIE INC 2016-04-27 CN disclosed