SCHEMBL28056901

SCHEMBL28056901

CC(C)(C)OC(=O)c1ccc(C(=O)N2CCc3ccccc3C2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 10/20 0.60
CYP3A4 P08684 2/20 0.60
CYP2C19 P33261 2/20 0.60
CYP2D6 P10635 1/20 0.60
HSP90AA1 P07900 2/20 0.59
HSP90AB1 P08238 2/20 0.59
LMNA P02545 1/20 0.57
CA1 P00915 1/20 0.57
CA2 P00918 1/20 0.57
CA7 P43166 1/20 0.57
CA9 Q16790 1/20 0.57
CA14 Q9ULX7 1/20 0.57
NAMPT P43490 1/20 0.57
TP53 P04637 2/20 0.56
ALDH1A1 P00352 6/20 0.54
SMN1; SMN2 Q16637 3/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
NOTUM Q6P988 1/20 0.52
HTT P42858 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31396757 0.84 NAMPT (0.68) HPGDHSP90AA1HSP90AB1LMNACA1
SCHEMBL14061184 0.84 HSP90AA1 (0.51) HPGDCYP3A4CYP2C19CYP2D6HSP90AA1
SCHEMBL3455632 0.82 HSP90AA1 (0.67) HPGDCYP3A4CYP2C19CYP2D6HSP90AA1
SCHEMBL14061114 0.82 HSP90AA1 (0.49) HPGDCYP3A4CYP2C19CYP2D6HSP90AA1
SCHEMBL28056773 0.82 MEN1 (0.72) HPGDCYP3A4CYP2C19CYP2D6LMNA
SCHEMBL13211911 0.80 HTT (0.71) HPGDCYP3A4CYP2C19CYP2D6HSP90AA1
SCHEMBL1202402 0.80 ESR2 (0.70) HPGDCYP3A4CYP2C19LMNANAMPT
SCHEMBL29369046 0.80 ESR2 (0.70) HPGDCYP3A4CYP2C19LMNANAMPT
SCHEMBL4279383 0.80 HPGD (0.73) HPGDCYP3A4CYP2C19CYP2D6LMNA
SCHEMBL30277860 0.80 HPGD (0.73) HPGDCYP3A4CYP2C19CYP2D6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103732589-B Can be used as the sulphonamide of the replacement of anti-apoptotic BCL inhibitor BRISTOL-MYERS SQUIBB CO. (US) 2016-03-30 CN disclosed