SCHEMBL28058825

SCHEMBL28058825

CC(C)C(=O)N1CCN(OC(=O)C(C)(C)C)C[C@H]1C

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAPT P10636 1/20 0.32
TSHR P16473 1/20 0.32
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28458593 0.82 TSHR (0.33) MAPTTSHRGAA
SCHEMBL17560452 0.73 SETD7 (0.47) SMN1; SMN2MAPT
SCHEMBL17560451 0.73 SETD7 (0.47) SMN1; SMN2MAPT
SCHEMBL23876834 0.73 PIK3CD (0.38) PIK3CDSMN1; SMN2MAPTTSHRGAA
SCHEMBL17589229 0.73 PIK3CD (0.38) PIK3CDSMN1; SMN2MAPTTSHRGAA
SCHEMBL28827116 0.71
SCHEMBL318016 0.71
SCHEMBL24368980 0.71 PIK3CD (0.41) PIK3CDSMN1; SMN2MAPTTSHRGAA
SCHEMBL23187990 0.71 PIK3CD (0.41) PIK3CDSMN1; SMN2MAPTTSHRGAA
SCHEMBL18346746 0.71 PIK3CD (0.41) PIK3CDSMN1; SMN2MAPTTSHRGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110088098-A Quinazolinones PARP-1 inhibitor and preparation method thereof, pharmaceutical composition and purposes 中国医学科学院药物研究所 2019-08-02 CN disclosed
CN-105461697-A Quinazolinone PARP-1 inhibitors, medicinal composition containing inhibitors, and antitumor use of inhibitors INST MATERIA MEDICA CAMS 2016-04-06 CN disclosed
CN-105399698-A Aromatic heterocyclic derivatives and applications of aromatic heterocyclic derivatives in medicines GUANGDONG HEC PHARMACEUTICAL 2016-03-16 CN disclosed