SCHEMBL28059226

SCHEMBL28059226

CC(=O)C1CNCCN1c1ccccn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLD1 Q13393 1/20 0.48
ALDH1A1 P00352 5/20 0.41
HPGD P15428 3/20 0.41
HSD17B10 Q99714 3/20 0.41
USP2 O75604 2/20 0.40
TSHR P16473 2/20 0.40
HIF1A Q16665 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
GRM1 Q13255 2/20 0.40
HTR2A P28223 4/20 0.40
HTR2C P28335 4/20 0.40
HTR2B P41595 4/20 0.40
ALOX5 P09917 1/20 0.40
MEN1 O00255 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29464840 0.88 PLD1 (0.49) PLD1ALDH1A1HPGDHSD17B10USP2
SCHEMBL9371314 0.83 GSK3B (0.42) GRM1HTR2AHTR2CHTR2B
SCHEMBL20141500 0.79 PLD1 (0.54) PLD1ALDH1A1HPGDHSD17B10USP2
SCHEMBL20129603 0.79 PLD1 (0.54) PLD1ALDH1A1HPGDHSD17B10USP2
SCHEMBL30531432 0.79 PLD1 (0.54) PLD1ALDH1A1HPGDHSD17B10USP2
SCHEMBL20129613 0.79 PLD1 (0.54) PLD1ALDH1A1HPGDHSD17B10USP2
SCHEMBL28059132 0.78 MMP1 (0.47) ALDH1A1HPGDHSD17B10USP2TSHR
Hydrochloric Acid SCHEMBL20141815 0.77 PLD1 (0.53) PLD1ALDH1A1HPGDHSD17B10USP2
Hydrochloric Acid SCHEMBL20141813 0.77 PLD1 (0.53) PLD1ALDH1A1HPGDHSD17B10USP2
SCHEMBL7262930 0.76 HTR2C (0.44) SMN1; SMN2HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107635986-A Substituted quinoxaline derivatives 赛尔维他股份公司 2018-01-26 CN claimed
CN-105814050-B Pyrazolopyridine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2018-05-08 CN disclosed
CN-105814059-B Imidazo pyrimidine derivatives as TNF active regulators UCB生物制药私人有限公司 2018-04-03 CN disclosed
CN-105814048-B Fused tricyclic benzimidizole derivatives as TNF active regulators UCB生物制药私人有限公司 2018-03-27 CN disclosed
CN-107787319-A Indazole derivatives as modulators of TNF activity UCB生物制药私人有限公司 2018-03-09 CN disclosed
CN-107690434-A Fused tricyclic Imidazopyrazines derivative as TNF active regulators UCB生物制药私人有限公司 2018-02-13 CN disclosed
CN-105814060-B Imidazo-triazine derivative as TNF active regulators UCB生物制药私人有限公司 2018-02-13 CN disclosed
CN-105814046-B Imidazopyridine derivatives as TNF active regulators UCB生物制药私人有限公司 2018-01-30 CN disclosed
CN-105814061-B Imidazopyridazine derivative as TNF active regulators UCB生物制药私人有限公司 2018-01-26 CN disclosed
CN-107635986-A Substituted quinoxaline derivatives 赛尔维他股份公司 2018-01-26 CN disclosed
CN-105814059-A Imidazopyrimidine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814050-A Pyrazolopyridine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814065-A Imidazothiazole derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814047-A Fused tricyclic benzimidazoles derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814051-A Tetrahydroimidazopyridine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814025-A Tetrahydrobenzimidazole derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814054-A Fused imidazole and pyrazole derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814049-A Fused tricyclic imidazole derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814043-A Triazolopyridine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814048-A Fused tricyclic imidazole derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed