SCHEMBL28059266

SCHEMBL28059266

C=CC(=O)Nc1cccc(Nc2ncc(Cl)c(Nc3cccc(NC(=O)C=C)c3)n2)c1

nearest known ligand 0.77

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EGFR P00533 14/20 0.77
BTK Q06187 7/20 0.71
ITK Q08881 2/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17936495 0.91 JAK3 (0.69) EGFRBTK
SCHEMBL9945478 0.90 BTK (0.67) EGFRBTK
SCHEMBL16513260 0.89 JAK3 (0.77) EGFRBTK
SCHEMBL28059285 0.89 EGFR (0.67) EGFRBTKITK
SCHEMBL29537933 0.89 JAK3 (0.77) EGFRBTK
SCHEMBL24392803 0.89 JAK3 (0.77) EGFRBTK
SCHEMBL16513364 0.88 EGFR (0.68) EGFRBTKITK
SCHEMBL9925321 0.88 EGFR (0.68) EGFRBTK
SCHEMBL16513456 0.87 EGFR (0.67) EGFRBTKITK
SCHEMBL16513279 0.86 JAK3 (0.66) EGFRBTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105384695-B Pyrimidine derivative, preparation method and medical application thereof 四川海思科制药有限公司 2019-12-20 CN disclosed
CN-105384695-A Pyrimidine derivative, preparation method therefor and application thereof in medicine SICHUAN HAISCO PHARMACEUTICAL CO LTD 2016-03-09 CN disclosed