SCHEMBL28059595

SCHEMBL28059595

O=Cc1cccc2cc(Br)oc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.46
CHRM4 P08173 1/20 0.46
CHRM5 P08912 1/20 0.46
CHRM1 P11229 1/20 0.46
CHRM3 P20309 1/20 0.46
TRIM24 O15164 2/20 0.41
TRIM33 Q9UPN9 2/20 0.41
ERN1 O75460 5/20 0.40
MEN1 O00255 2/20 0.38
THRB P10828 2/20 0.38
KMT2A Q03164 2/20 0.38
LMNA P02545 1/20 0.38
BLM P54132 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CYP2A6 P11509 2/20 0.38
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
ALDH1A1 P00352 3/20 0.34
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8082599 0.78 CHRM2 (0.46) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL28066198 0.75 TYR (0.51) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL8678236 0.74 MAOA (0.58) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL28190803 0.74 CHRM2 (0.43) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL28045400 0.73 CHRM2 (0.45) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL971239 0.72 CYP2A6 (0.51) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL21797929 0.71 AHR (0.39) MEN1KMT2ACYP2A6ALDH1A1HPGD
Hydrochloric Acid SCHEMBL14686366 0.70 CYP2A6 (0.50) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL31033079 0.69 MAOB (0.55) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL1802080 0.67 MEN1 (0.42) CHRM2CHRM4CHRM5CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105492437-A Substituted benzofuranyl and benzoxazolyl compounds and uses thereof KARYOPHARM THERAPEUTICS INC 2016-04-13 CN disclosed