SCHEMBL28059708

SCHEMBL28059708

CCC(C(=O)O)c1ccc(F)c(F)c1F

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.45
CES1 P23141 2/20 0.45
AKR1C3 P42330 11/20 0.42
AKR1C2 P52895 11/20 0.42
AKR1C1 Q04828 2/20 0.36
AKR1B10 O60218 1/20 0.36
AKR1C4 P17516 1/20 0.36
PTGS1 P23219 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5153327 0.83 AKR1C3 (0.38) AKR1C3AKR1C2AKR1C1PTGS1
SCHEMBL1343470 0.78 CYP1A2 (0.44) AKR1C3AKR1C2
SCHEMBL16963923 0.77 CES2 (0.46) CES2CES1AKR1C3AKR1C2AKR1C1
SCHEMBL27934340 0.77 CES2 (0.41) CES2CES1
SCHEMBL1966206 0.76 KCNQ2 (0.49) CES2CES1AKR1C3AKR1C2AKR1C1
SCHEMBL30427742 0.76 KCNQ2 (0.49) CES2CES1AKR1C3AKR1C2AKR1C1
SCHEMBL154992 0.76 AKR1C3 (0.40) AKR1C3AKR1C2AKR1C1AKR1B10AKR1C4
SCHEMBL19200334 0.76 AKR1C3 (0.50) AKR1C3AKR1C2AKR1C1AKR1B10AKR1C4
SCHEMBL909711 0.76 AKR1C3 (0.40) AKR1C3AKR1C2AKR1C1AKR1B10AKR1C4
SCHEMBL23412757 0.76 CES2 (0.40) CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103172539-B The preparation method of Glucovance sitagliptin intermediate aminobenzene butyric acid derivative 上海阳帆医药科技有限公司 2016-08-03 CN disclosed