SCHEMBL28060087

SCHEMBL28060087

COc1cccc(Nc2nc(-c3ccc(C4CCC(CCOC(C)=O)CC4)cc3)cs2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 10/20 0.57
KMT2A Q03164 10/20 0.57
NPC1 O15118 6/20 0.57
MAPT P10636 6/20 0.57
CYP1A2 P05177 3/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C9 P11712 1/20 0.57
PKM P14618 1/20 0.57
CYP2C19 P33261 1/20 0.57
CLK1 P49759 1/20 0.57
GSK3A P49840 1/20 0.57
GSK3B P49841 1/20 0.57
CDK5 Q00535 1/20 0.57
CDK5R1 Q15078 1/20 0.57
PTGS2 P35354 3/20 0.55
RAB9A P51151 6/20 0.52
ALDH1A1 P00352 4/20 0.52
SMN1; SMN2 Q16637 4/20 0.52
GAA P10253 3/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL180959 0.86 MEN1 (0.61) MEN1KMT2ANPC1MAPTCYP1A2
SCHEMBL13664061 0.86 MEN1 (0.61) MEN1KMT2ANPC1MAPTCYP1A2
SCHEMBL14617023 0.86 MEN1 (0.61) MEN1KMT2ANPC1MAPTCYP1A2
SCHEMBL1722325 0.86 MEN1 (0.61) MEN1KMT2ANPC1MAPTCYP1A2
SCHEMBL27790830 0.86 MEN1 (0.63) MEN1KMT2ANPC1MAPTCYP1A2
SCHEMBL180876 0.85 MEN1 (0.57) MEN1KMT2ANPC1MAPTCYP1A2
SCHEMBL28060088 0.83 MEN1 (0.59) MEN1KMT2ANPC1MAPTCYP1A2
SCHEMBL27769454 0.81 MEN1 (0.67) MEN1KMT2ANPC1MAPTCYP1A2
SCHEMBL27769395 0.76 ALOX5 (0.56) MEN1KMT2ANPC1MAPTCYP1A2
SCHEMBL12297791 0.75 MEN1 (0.84) MEN1KMT2ANPC1MAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103288721-B (4-(4-[6-(trifluoromethylpyridin-3-base amino)-containing N heteroaryl]-phenyl)-cyclohexyl)-acetogenin and pharmaceutical use thereof NOVARTIS AG (CH) 2016-04-20 CN disclosed