SCHEMBL28060123

SCHEMBL28060123

C#Cc1cc(OC)ccc1F

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.41
FBP1 P09467 1/20 0.41
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA7 P43166 2/20 0.39
CA9 Q16790 2/20 0.39
CA14 Q9ULX7 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP1A1 P04798 1/20 0.39
CYP1B1 Q16678 1/20 0.39
CYP2A6 P11509 1/20 0.38
NFE2L2 Q16236 1/20 0.38
MTNR1B P49286 2/20 0.37
CPS1 P31327 1/20 0.37
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2720566 0.84 CYP1A2 (0.42) CA12CA1CA2CA7CA9
SCHEMBL29641932 0.84 CYP1A2 (0.42) CA12CA1CA2CA7CA9
SCHEMBL1017145 0.80 CYP11B1 (0.47)
SCHEMBL30079514 0.80 CYP11B1 (0.47)
SCHEMBL6212996 0.80 CPS1 (0.40) CA12CA1CA2CA7CA9
SCHEMBL16959354 0.80 CA12 (0.39) CA12CA1CA2CA7CA9
SCHEMBL31119234 0.78 CA12 (0.56) CA12CA1CA2CA7CA9
SCHEMBL6196567 0.78 CA12 (0.56) CA12CA1CA2CA7CA9
SCHEMBL29870653 0.77 GPR3 (0.42) CYP1A2
SCHEMBL26426439 0.77 GPR3 (0.42) CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105492429-A Heteroaryl inhibitors of SUMO activating enzyme MILLENNIUM PHARM INC 2016-04-13 CN disclosed