SCHEMBL280628

SCHEMBL280628

Fc1ccc([C@@H]2COCCN2)cc1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CSNK1D P48730 1/20 0.43
CSNK1E P49674 1/20 0.43
KCNH2 Q12809 1/20 0.43
PRKACA P17612 1/20 0.41
PRKACG P22612 1/20 0.41
PRKACB P22694 1/20 0.41
TACR1 P25103 8/20 0.40
ACVR1 Q04771 1/20 0.39
PRCP P42785 1/20 0.37
CTSK P43235 1/20 0.35
KDM1A O60341 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18387 1.00 CSNK1D (0.43) CSNK1DCSNK1EKCNH2PRKACAPRKACG
SCHEMBL8321907 1.00 CSNK1D (0.43) CSNK1DCSNK1EKCNH2PRKACAPRKACG
Hydrochloric Acid SCHEMBL28500586 0.98 CSNK1D (0.43) CSNK1DCSNK1EKCNH2PRKACAPRKACG
Hydrochloric Acid SCHEMBL28214300 0.98 CSNK1D (0.43) CSNK1DCSNK1EKCNH2PRKACAPRKACG
SCHEMBL2944138 0.81 CHRNA7 (0.47) PRKACAPRKACGPRKACBPRCPCTSK
SCHEMBL3399522 0.81 PRKACA (0.47) CSNK1DCSNK1EKCNH2PRKACAPRKACG
SCHEMBL14839620 0.81 PRKACA (0.41) PRKACAPRKACGPRKACBACVR1CTSK
SCHEMBL22589151 0.81 CHRNA7 (0.47) PRKACAPRKACGPRKACBPRCPCTSK
SCHEMBL21717791 0.81 MAPT (0.44) KCNH2PRKACAPRKACGPRKACBACVR1
SCHEMBL5545595 0.81 MAPT (0.44) CSNK1DCSNK1EKCNH2PRKACAPRKACG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8133994-B2 Preparation of aprepitant DR. REDDY'S LABORATORIES LTD. (IN) 2012-03-13 US disclosed
US-20110094321-A1 PREPARATION OF APREPITANT DR. REDDY'S LABORATORIES LIMITED (IN) 2011-04-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110094321-A1 PREPARATION OF APREPITANT KIT, CPA3, CMA1 CSNK1D 1489/4885CSNK1E 943/4885KCNH2 1289/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.