SCHEMBL28064690

SCHEMBL28064690

NC1=NC=C(C(F)(F)F)C(N)(c2cccc([N+](=O)[O-])c2)N1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.42
ALDH1A1 P00352 1/20 0.38
LMNA P02545 3/20 0.36
TSHR P16473 1/20 0.36
BACE1 P56817 1/20 0.36
CHRNA1 P02708 1/20 0.36
CHRNG P07510 1/20 0.36
CHRNB1 P11230 1/20 0.36
CHRNB2 P17787 1/20 0.36
SLC6A2 P23975 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
SLC6A3 Q01959 1/20 0.36
CHRND Q07001 1/20 0.36
NFE2L2 Q16236 2/20 0.35
TDO2 P48775 1/20 0.35
MAPT P10636 1/20 0.35
NPY5R Q15761 1/20 0.35
CYP19A1 P11511 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28064702 0.82 CHRNA1 (0.43) KDM1AALDH1A1LMNATSHRCHRNA1
SCHEMBL30764023 0.78 GRM4 (0.33) ALDH1A1TSHRBACE1
SCHEMBL28064648 0.72 KDM1A (0.44) KDM1AALDH1A1LMNATSHRCHRNA1
SCHEMBL18007509 0.66 KDM1A (0.51) KDM1AALDH1A1LMNATSHRCHRNA1
SCHEMBL18007717 0.66 KDM1A (0.55) KDM1AALDH1A1LMNATSHRGAA
SCHEMBL29703748 0.64 TSHR (0.61) ALDH1A1LMNATSHRNFE2L2MAPT
SCHEMBL439710 0.64 TSHR (0.61) ALDH1A1LMNATSHRNFE2L2MAPT
SCHEMBL9848305 0.63 KDM1A (0.59) KDM1AALDH1A1LMNATSHRNFE2L2
SCHEMBL24027901 0.63 KDM1A (0.55) KDM1AALDH1A1LMNATSHRCHRNA1
SCHEMBL29203888 0.63 KIF11 (0.59) ALDH1A1LMNATSHRNFE2L2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105503827-A EGFR (Epidermal growth factor receptor) inhibitor and preparation method and use thereof SHANGHAI HANSOH BIOMEDICAL CO LTD 2016-04-20 CN disclosed