SCHEMBL28064867

SCHEMBL28064867

O=[SH](=O)Cc1ccc(C2CCCCN2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C19 P33261 2/20 0.44
KMT2A Q03164 2/20 0.44
CHRNB2 P17787 2/20 0.44
CHRNA7 P36544 2/20 0.44
CHRNA4 P43681 2/20 0.44
POLB P06746 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2A6 P11509 1/20 0.44
CYP2C9 P11712 1/20 0.44
AURKA O14965 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
MKNK1 Q9BUB5 1/20 0.38
PARP1 P09874 3/20 0.37
PARP2 Q9UGN5 2/20 0.37
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
MAPKAPK2 P49137 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1652841 0.81 MEN1 (0.47) MEN1CYP2D6CYP2C19KMT2ACHRNB2
SCHEMBL8611268 0.81 CYP2D6 (0.47) MEN1CYP2D6CYP2C19KMT2ACHRNB2
SCHEMBL27351589 0.78 MEN1 (0.47) MEN1CYP2D6CYP2C19KMT2ACHRNB2
SCHEMBL716893 0.76 MKNK1 (0.48) MEN1CYP2D6CYP2C19KMT2ACHRNB2
SCHEMBL6178200 0.76 MKNK1 (0.48) MEN1CYP2D6CYP2C19KMT2ACHRNB2
SCHEMBL23891896 0.74 CYP2D6 (0.44) MEN1CYP2D6CYP2C19KMT2ACHRNB2
SCHEMBL21806676 0.73 CHRNB2 (0.44) MEN1CYP2D6CYP2C19KMT2ACHRNB2
SCHEMBL16409303 0.73 CYP4F2 (0.46) MEN1CYP2D6CYP2C19KMT2ACHRNB2
SCHEMBL13499189 0.72 HRH3 (0.55) MEN1CYP2D6CYP2C19KMT2APOLB
SCHEMBL3081329 0.72 MEN1 (0.51) MEN1CYP2D6CYP2C19KMT2ACHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105579444-B Piperidinylindole derivatives and their use as complement factor B inhibitors 诺华股份有限公司 2018-05-01 CN disclosed
CN-105579444-A Piperidinylindole derivatives and their use as complement factor B inhibitors NOVARTIS AG 2016-05-11 CN disclosed