SCHEMBL28065241

SCHEMBL28065241

O=C(O)CCNC(=O)c1csc(-c2cccc(Cl)c2Cl)n1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PANK3 Q9H999 1/20 0.72
TLR7 Q9NYK1 1/20 0.61
HTR2C P28335 5/20 0.52
LMNA P02545 3/20 0.45
HPGD P15428 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
RXRA P19793 1/20 0.42
RXRB P28702 1/20 0.42
RXRG P48443 1/20 0.42
TDP1 Q9NUW8 2/20 0.42
MAPT P10636 3/20 0.42
ALDH1A1 P00352 2/20 0.42
ATM Q13315 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7549240 0.83 PANK3 (0.71) PANK3TLR7HTR2CHPGDHDAC3
SCHEMBL28065290 0.81 CYP1A2 (0.49) PANK3LMNAHPGDCYP1A2CYP3A4
SCHEMBL27966313 0.81 HIF1A (0.52) PANK3LMNAHPGDCYP1A2CYP3A4
SCHEMBL3537090 0.80 PANK3 (0.64) PANK3TLR7HTR2CNPSR1L3MBTL1
SCHEMBL27966332 0.80 HPGD (0.66) TLR7LMNAHPGDCYP1A2CYP3A4
SCHEMBL3538271 0.79 HTR2C (0.64) PANK3TLR7HTR2CALDH1A1KDM4E
SCHEMBL14716946 0.79 PANK3 (0.62) PANK3TLR7HTR2CLMNAHPGD
SCHEMBL14662725 0.77 CTSA (0.66) PANK3TLR7
SCHEMBL14662722 0.77 CTSA (0.66) PANK3TLR7
SCHEMBL3539520 0.76 HTR2C (0.64) PANK3TLR7HTR2CKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103827098-B The 3-(thiazole-4-carbonyl)-replaced or 3-(thiazole-2-carbonyl)-alanine derivatives and the purposes as medicine thereof 赛诺菲 2016-06-15 CN claimed
CN-103827098-B The 3-(thiazole-4-carbonyl)-replaced or 3-(thiazole-2-carbonyl)-alanine derivatives and the purposes as medicine thereof 赛诺菲 2016-06-15 CN disclosed