Choline

Choline

SCHEMBL28067091

C[N+](C)(C)CCO.O=C(O)C(F)(F)F

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADORA1ADORA2AADORA2BADORA3GNRHRMPLPDE3APDE3BPDE4APDE4BPDE4CPDE4DPPARASLC5A2

The experimentally established mechanism targets of Choline. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.55
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
CYP3A4 P08684 1/20 0.55
SLC5A7 Q9GZV3 1/20 0.55
TSHR P16473 2/20 0.35
ACHE P22303 1/20 0.34
CHRM5 P08912 4/20 0.33
CHRM1 P11229 4/20 0.33
CHRM3 P20309 4/20 0.33
CHRM2 P08172 3/20 0.33
CHRM4 P08173 3/20 0.33
CYP2C19 P33261 3/20 0.33
GALR3 O60755 2/20 0.33
HTR1A P08908 2/20 0.33
CHRNB2 P17787 2/20 0.33
CHRNA7 P36544 2/20 0.33
CHRNA4 P43681 2/20 0.33
ADRA2A P08913 1/20 0.33
ADRA1A P35348 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Choline SCHEMBL28566318 0.98 CYP3A4 (0.59) LMNAMEN1KMT2ACYP3A4SLC5A7
Choline SCHEMBL3784402 0.84 LMNA (0.52) LMNAMEN1KMT2ACYP3A4SLC5A7
Pivalate SCHEMBL27641475 0.83 LMNA (0.57) LMNAMEN1KMT2ACYP3A4SLC5A7
Choline SCHEMBL15993849 0.82 CYP3A4 (0.56) LMNAMEN1KMT2ACYP3A4SLC5A7
Choline SCHEMBL15993791 0.82 LMNA (0.56) LMNAMEN1KMT2ACYP3A4SLC5A7
Choline SCHEMBL15994029 0.82 LMNA (0.50) LMNAMEN1KMT2ACYP3A4SLC5A7
Choline SCHEMBL15994026 0.82 CYP3A4 (0.56) LMNAMEN1KMT2ACYP3A4SLC5A7
Choline SCHEMBL15993799 0.82 CYP3A4 (0.56) LMNAMEN1KMT2ACYP3A4SLC5A7
Choline SCHEMBL2445125 0.82 LMNA (0.71) LMNAMEN1KMT2ACYP3A4SLC5A7
Choline SCHEMBL15993937 0.80 CYP3A4 (0.54) LMNAMEN1KMT2ACYP3A4SLC5A7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105503540-A Method for preparation of benzene ring phenol compound from alkali lignin DALIAN INST CHEMICAL PHYSICS CAS 2016-04-20 CN claimed
CN-105503540-A Method for preparation of benzene ring phenol compound from alkali lignin DALIAN INST CHEMICAL PHYSICS CAS 2016-04-20 CN disclosed