SCHEMBL28067941

SCHEMBL28067941

c1ccc(Cc2cncn2C(c2ccccc2)(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 4/20 0.42
CYP11B2 P19099 4/20 0.42
IDO1 P14902 1/20 0.36
CALM1 P0DP23 1/20 0.35
P2RX7 Q99572 1/20 0.35
CYP19A1 P11511 2/20 0.35
TAAR1 Q96RJ0 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
HIF1A Q16665 2/20 0.35
KCNA5 P22460 1/20 0.35
LMNA P02545 2/20 0.35
MEN1 O00255 1/20 0.35
SLC22A1 O15245 1/20 0.35
KCNN4 O15554 1/20 0.35
NR1I2 O75469 1/20 0.35
GMNN O75496 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8481796 0.81 CYP11B1 (0.40) CYP11B1CYP11B2IDO1CYP19A1CYP1A2
SCHEMBL1765841 0.81 CYP11B1 (0.40) CYP11B1CYP11B2P2RX7CYP19A1CYP1A2
SCHEMBL25307807 0.79 CYP11B1 (0.38) CYP11B1CYP11B2TAAR1NR1I2ADORA3
SCHEMBL27579878 0.79 CYP11B1 (0.38) CYP11B1CYP11B2CYP19A1CYP1A2CYP3A4
SCHEMBL9235495 0.78 CYP11B1 (0.37) CYP11B1CYP11B2CYP19A1CYP1A2CYP3A4
SCHEMBL10818578 0.78 CYP11B1 (0.37) CYP11B1CYP11B2IDO1CYP19A1CYP1A2
SCHEMBL25368193 0.78 CYP11B1 (0.37) CYP11B1CYP11B2IDO1CYP19A1CYP1A2
SCHEMBL6613495 0.78 HDAC3 (0.40) CYP11B1CYP11B2CYP2C19HIF1ATBXAS1
SCHEMBL9239487 0.78 CYP11B1 (0.37) CYP11B1CYP11B2CYP19A1CYP1A2CYP3A4
SCHEMBL6978240 0.77 CYP11B1 (0.37) CYP11B1CYP11B2IDO1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108864102-A ERK inhibitor and application method 库拉肿瘤学公司 2018-11-23 CN disclosed
CN-105636586-B ERK inhibitors and methods of use 库拉肿瘤学公司 2018-05-29 CN disclosed
CN-105636586-A ERK inhibitors and methods of use ARAXES PHARMA LLC 2016-06-01 CN disclosed