SCHEMBL28068161

SCHEMBL28068161

COc1cc(C(=O)N2CCCC2CO)c(NC(=O)O)cc1O

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.45
TRPV1 Q8NER1 2/20 0.43
TLR8 Q9NR97 1/20 0.42
TLR7 Q9NYK1 1/20 0.42
HCRTR1 O43613 3/20 0.40
HCRTR2 O43614 3/20 0.40
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.39
SPHK2 Q9NRA0 1/20 0.39
LRRK2 Q5S007 1/20 0.38
DRD2 P14416 1/20 0.38
POLB P06746 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28439902 1.00 ROCK2 (0.45) ROCK2TRPV1TLR8TLR7HCRTR1
SCHEMBL20975315 0.97 TRPV1 (0.44) ROCK2TRPV1TLR8TLR7HCRTR1
SCHEMBL20975319 0.97 TRPV1 (0.44) ROCK2TRPV1TLR8TLR7HCRTR1
SCHEMBL16781580 0.87 ROCK2 (0.42) ROCK2TRPV1TLR8TLR7HCRTR1
SCHEMBL16486542 0.87 ROCK2 (0.42) ROCK2TRPV1TLR8TLR7HCRTR1
SCHEMBL28068160 0.85 ROCK2 (0.45) ROCK2TRPV1TLR8TLR7HCRTR1
SCHEMBL30944529 0.84 TRPV1 (0.41) ROCK2TRPV1TLR8TLR7HCRTR1
SCHEMBL4413990 0.84 ROCK2 (0.47) ROCK2TRPV1TLR8TLR7HCRTR1
SCHEMBL13594838 0.84 ROCK2 (0.47) ROCK2TRPV1TLR8TLR7HCRTR1
SCHEMBL16486649 0.82 ROCK2 (0.48) ROCK2TRPV1TLR8TLR7HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105636612-A 1- (chloromethyl) -2, 3-dihydro-1H-benzo [ e ] indole dimer antibody-drug conjugate compounds, and methods of use and treatment GENENTECH INC 2016-06-01 CN disclosed