SCHEMBL28068959

SCHEMBL28068959

Cc1ccc(Sc2nc3c(N)ncnc3[nH]2)c(C)c1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.38
HSP90AB1 P08238 2/20 0.38
ERBB2 P04626 1/20 0.38
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36
NUDT1 P36639 1/20 0.35
MAP4K4 O95819 5/20 0.34
KDM4E B2RXH2 1/20 0.33
PIK3CD O00329 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33
PIK3CG P48736 1/20 0.33
PRKDC P78527 1/20 0.33
PI4KA P42356 3/20 0.32
PI4K2B Q8TCG2 3/20 0.32
PI4K2A Q9BTU6 3/20 0.32
PI4KB Q9UBF8 3/20 0.32
HSP90B1 P14625 2/20 0.32
TRAP1 Q12931 1/20 0.32
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16487461 0.83 HSP90B1 (0.47) HSP90AA1HSP90AB1ERBB2LMNATSHR
SCHEMBL11980432 0.82 MAP4K4 (0.42) HSP90AA1HSP90AB1ERBB2LMNATSHR
SCHEMBL13050401 0.81 HSP90AA1 (0.42) HSP90AA1HSP90AB1ERBB2LMNATSHR
SCHEMBL14467034 0.79 ERBB2 (0.41) HSP90AA1HSP90AB1ERBB2MAP4K4
SCHEMBL3517738 0.77 HSP90AA1 (0.40) HSP90AA1HSP90AB1ERBB2LMNATSHR
SCHEMBL1669646 0.76 ERBB2 (0.40) HSP90AA1HSP90AB1ERBB2LMNATSHR
SCHEMBL16486623 0.76 HSP90AA1 (0.46) HSP90AA1HSP90AB1ERBB2LMNATSHR
SCHEMBL15080556 0.75 HSP90AA1 (0.49) HSP90AA1HSP90AB1ERBB2LMNATSHR
SCHEMBL16486451 0.75 HSP90B1 (0.44) HSP90AA1HSP90AB1ERBB2LMNATSHR
SCHEMBL3124207 0.75 LMNA (0.36) HSP90AA1HSP90AB1ERBB2LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105899503-B Selective GRP94 inhibitors and uses thereof 纪念斯隆-凯特琳癌症中心 2020-08-18 CN disclosed
CN-105899503-A Selective GRP94 inhibitors and uses thereof 纪念斯隆-凯特琳癌症中心 2016-08-24 CN disclosed