Quinoline

Quinoline

SCHEMBL28069084

Brc1cc2cccnc2[nH]1.c1ccc2ncccc2c1

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.57
HTT P42858 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C19 P33261 1/20 0.47
RIPK1 Q13546 9/20 0.45
DAO P14920 1/20 0.45
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
POLB P06746 1/20 0.42
CCNB2 O95067 1/20 0.40
CDK1 P06493 1/20 0.40
CCNB1 P14635 1/20 0.40
CCNB3 Q8WWL7 1/20 0.40
CASP1 P29466 2/20 0.40
MEN1 O00255 1/20 0.40
CASP7 P55210 1/20 0.40
KMT2A Q03164 1/20 0.40
NR4A2 P43354 1/20 0.40
KDM4E B2RXH2 1/20 0.40
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2595303 0.89 DAO (0.53) RIPK1DAOCCNB2CDK1CCNB1
Quinoline SCHEMBL28065955 0.83 ALDH1A1 (0.57) ALDH1A1HTTCYP1A2CYP2C19NPC1
Quinoline SCHEMBL27928312 0.80 ALDH1A1 (0.49) ALDH1A1HTTCYP1A2CYP2C19DAO
Quinoline SCHEMBL28216931 0.80 ALDH1A1 (0.57) ALDH1A1HTTCYP1A2CYP2C19RIPK1
Quinoline SCHEMBL137291 0.78 ALDH1A1 (0.94) ALDH1A1HTTCYP1A2CYP2C19NPC1
Quinoline SCHEMBL27611581 0.75 ALDH1A1 (0.90) ALDH1A1HTTCYP1A2CYP2C19NPC1
Quinoline SCHEMBL27594824 0.75 ALDH1A1 (0.90) ALDH1A1HTTCYP1A2CYP2C19NPC1
Quinoline SCHEMBL29349552 0.75 ALDH1A1 (1.00) ALDH1A1HTTCYP1A2CYP2C19NPC1
Quinoline SCHEMBL32661377 0.75 ALDH1A1 (1.00) ALDH1A1HTTCYP1A2CYP2C19NPC1
Quinoline SCHEMBL29822171 0.75 ALDH1A1 (1.00) ALDH1A1HTTCYP1A2CYP2C19NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105622605-A Synthesis method of 5-bromo-7-azaindole ITIC MEDCHEM CO LTD 2016-06-01 CN claimed
CN-105622605-A Synthesis method of 5-bromo-7-azaindole ITIC MEDCHEM CO LTD 2016-06-01 CN disclosed