SCHEMBL28069576

SCHEMBL28069576

Cn1c(=O)cc(N2CCC[C@@H](C(=O)OC(C)(C)C)C2N)n(Cc2cc(F)ccc2C#N)c1=O

nearest known ligand 0.62

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 20/20 0.62
OPRM1 P35372 1/20 0.47
OPRK1 P41145 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28507241 0.80 DPP4 (0.59) DPP4OPRM1OPRK1CYP1A2CYP3A4
SCHEMBL28507242 0.78 DPP4 (0.68) DPP4OPRM1OPRK1CYP1A2CYP3A4
SCHEMBL28069573 0.78 DPP4 (0.68) DPP4OPRM1OPRK1CYP1A2CYP3A4
Trelagliptin SCHEMBL175726 0.77 DPP4 (1.00) DPP4OPRM1OPRK1CYP1A2CYP3A4
Trelagliptin SCHEMBL29349599 0.77 DPP4 (1.00) DPP4OPRM1OPRK1CYP1A2CYP3A4
Trelagliptin SCHEMBL175727 0.77 DPP4 (1.00) DPP4OPRM1OPRK1CYP1A2CYP3A4
Trelagliptin SCHEMBL878010 0.75 DPP4 (1.00) DPP4OPRM1OPRK1CYP1A2CYP3A4
Trelagliptin SCHEMBL29364762 0.75 DPP4 (1.00) DPP4OPRM1OPRK1CYP1A2CYP3A4
Trelagliptin SCHEMBL19534887 0.75 DPP4 (1.00) DPP4OPRM1OPRK1CYP1A2CYP3A4
Trelagliptin SCHEMBL28390472 0.75 DPP4 (1.00) DPP4OPRM1OPRK1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105646447-A Synthesis method of dipeptidyl peptidase inhibitor 北京康立生医药技术开发有限公司 2016-06-08 CN disclosed