SCHEMBL28069849

SCHEMBL28069849

COc1cccc2c1CCC2C(=O)C1CCc2c(OC)cccc21

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 2/20 0.54
DRD4 P21917 3/20 0.50
DRD2 P14416 3/20 0.50
DRD3 P35462 3/20 0.50
MEN1 O00255 2/20 0.50
CYP1A2 P05177 2/20 0.50
HTR1A P08908 2/20 0.50
HTR5A P47898 2/20 0.50
KMT2A Q03164 2/20 0.50
CYP2D6 P10635 1/20 0.50
CYP19A1 P11511 1/20 0.49
HSD11B1 P28845 1/20 0.49
MTNR1A P48039 2/20 0.48
MTNR1B P49286 2/20 0.48
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
KDM4E B2RXH2 1/20 0.47
LMNA P02545 1/20 0.47
POLB P06746 1/20 0.47
MAPT P10636 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1847083 0.89 PIN1 (0.52) PIN1DRD4DRD2DRD3MEN1
SCHEMBL20478665 0.89 PIN1 (0.52) PIN1DRD4DRD2DRD3MEN1
SCHEMBL20478637 0.88 PIN1 (0.51) PIN1DRD4DRD2DRD3MEN1
SCHEMBL12662601 0.80 CA1 (0.53) PIN1DRD4CA1CA2TAS1R3
SCHEMBL9325738 0.80 CA1 (0.53) DRD4CA1CA2TAS1R3TAS1R1
SCHEMBL1844443 0.80 CA1 (0.53) DRD4CA1CA2TAS1R3TAS1R1
SCHEMBL5848209 0.79 CA1 (0.55) DRD4CA1CA2TAS1R3TAS1R1
SCHEMBL20478894 0.79 CA1 (0.52) PIN1DRD4CA1CA2TAS1R3
SCHEMBL5848210 0.79 CA1 (0.55) DRD4CA1CA2TAS1R3TAS1R1
SCHEMBL5520518 0.79 CA1 (0.55) PIN1DRD4CA1CA2TAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110372550-A Aryl ether and application thereof 佩洛通治疗公司 2019-10-25 CN disclosed
CN-105530923-B Aryl ethers and their use 佩洛通治疗公司 2019-07-23 CN disclosed
CN-105530923-A Aryl ethers and their use PELOTON THERAPEUTICS INC 2016-04-27 CN disclosed